SCHEMBL4638260

SCHEMBL4638260

C#CCOc1ccc(C=O)c(F)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GSTP1 P09211 1/20 0.45
CA12 O43570 6/20 0.43
CA4 P22748 6/20 0.43
CA9 Q16790 6/20 0.43
CA1 P00915 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
TSHR P16473 1/20 0.43
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
MAOB P27338 6/20 0.41
KAT6A Q92794 1/20 0.40
MAOA P21397 3/20 0.39
ACHE P22303 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14117097 0.81 ADAM17 (0.40) ALDH1A1
SCHEMBL2024267 0.81 MAOB (0.45) GSTP1CA12CA4CA9CA1
SCHEMBL9636031 0.81 TYR (0.56) GSTP1CA12CA4CA9CA1
SCHEMBL17848287 0.80 GSTP1 (0.42) GSTP1CA12CA4CA9CA1
SCHEMBL18761828 0.79 GSTP1 (0.49) GSTP1CA12CA4CA9CA1
SCHEMBL9634543 0.78 ALDH1A1 (0.63) GSTP1CA12CA4CA9CA1
SCHEMBL3170130 0.78 NQO1 (0.45) KDM4EALDH1A1GAATSHR
SCHEMBL22322029 0.78 ALDH1A1 (0.37) ALDH1A1MAOBMAOA
SCHEMBL15080749 0.77 KDM4E (0.52) GSTP1CA12CA4CA9CA1
SCHEMBL14149542 0.77 MAOB (0.45) GSTP1CA12CA4CA9CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008099020-A1 1,1-DIOXO-1-THIA-5,10-DIAZADIBENZOCYCLOHEPTENES USEFUL AS HEPATITIS C VIRUS INHIBITORS TIBOTEC PHARMACEUTICALS LTD. (IE) 2008-08-21 WO disclosed
EP-1940780-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL CO., LTD. (JP) 2008-07-09 EP disclosed
EP-1940779-A2 AMIDE COMPOUNDS AND THEIR USE Sumitomo Chemical Company, Limited (JP) 2008-07-09 EP disclosed
WO-2007049729-A2 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-03 WO disclosed
WO-2007049728-A1 AMIDE COMPOUNDS AND THEIR USE SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2007-05-03 WO disclosed