SCHEMBL4637734

SCHEMBL4637734

COC(=O)c1nnn(Cc2ccc(F)c(F)c2)c1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 9/20 0.46
CYP1A2 P05177 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
PTGER4 P35408 1/20 0.41
FGFR1 P11362 1/20 0.40
FGFR4 P22455 1/20 0.40
IDH1 O75874 1/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
GABRA1 P14867 1/20 0.39
GABRG2 P18507 1/20 0.39
GABRB3 P28472 1/20 0.39
GABRA3 P34903 1/20 0.39
GABRA2 P47869 1/20 0.39
ALDH1A1 P00352 1/20 0.39
GRIN1 Q05586 1/20 0.38
GRIN2B Q13224 1/20 0.38
MAPK10 P53779 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637702 0.88 PTGER4 (0.44) CYP19A1PTGER4IDH1ALDH1A1GRIN1
SCHEMBL4637975 0.87 CYP19A1 (0.39) CYP19A1PTGER4IDH1ALDH1A1GRIN1
SCHEMBL4637971 0.86 CYP19A1 (0.50) CYP19A1CYP1A2SMN1; SMN2IDH1CYP11B1
SCHEMBL4638568 0.85 IDH1 (0.54) CYP19A1CYP1A2SMN1; SMN2PTGER4IDH1
SCHEMBL4637730 0.83 MAPT (0.50) CYP19A1CYP1A2SMN1; SMN2PTGER4IDH1
SCHEMBL4637999 0.83 IDH1 (0.46) CYP19A1CYP1A2SMN1; SMN2FGFR1IDH1
SCHEMBL4638905 0.77 IDH1 (0.41) CYP19A1SMN1; SMN2PTGER4IDH1ALDH1A1
SCHEMBL4637961 0.77 CFTR (0.46) CYP19A1SMN1; SMN2IDH1CYP11B1CYP11B2
SCHEMBL4637833 0.74 CYP19A1 (0.59) CYP19A1SMN1; SMN2IDH1GABRA1ALDH1A1
SCHEMBL23294412 0.73 MEN1 (0.49) CYP19A1CYP1A2SMN1; SMN2ALDH1A1GRIN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed