SCHEMBL4638728

SCHEMBL4638728

O=C(O)C1CN(c2ccc(F)c(F)c2)C(=O)O1

nearest known ligand 0.57

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.57
MAOA P21397 5/20 0.55
CALML3 P27482 6/20 0.44
BPTF Q12830 1/20 0.44
MAOB P27338 5/20 0.42
LMNA P02545 1/20 0.42
PTGS1 P23219 1/20 0.42
SDHA P31040 1/20 0.42
FADS1 O60427 1/20 0.40
F10 P00742 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638720 1.00 TSHR (0.57) TSHRMAOACALML3BPTFMAOB
SCHEMBL1224895 0.88 MAOA (0.52) TSHRMAOACALML3MAOBLMNA
SCHEMBL5763989 0.88 MAOA (0.52) TSHRMAOACALML3MAOBLMNA
SCHEMBL1224894 0.88 MAOA (0.52) TSHRMAOACALML3MAOBLMNA
SCHEMBL4757201 0.82 MAOA (0.61) TSHRMAOACALML3MAOBLMNA
SCHEMBL4637383 0.82 FADS1 (0.60) MAOAMAOBLMNAFADS1
SCHEMBL4637380 0.82 FADS1 (0.60) MAOAMAOBLMNAFADS1
SCHEMBL3038562 0.81 MAOB (0.65) TSHRMAOACALML3MAOBLMNA
SCHEMBL4757260 0.81 MAOB (0.47) MAOACALML3MAOBLMNAPTGS1
SCHEMBL6616635 0.81 MAOB (0.66) MAOACALML3MAOBLMNAPTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1937655-A1 HIV-1 PROTEASE INHIBITORS, AND METHODS OF MAKING AND USING THEM University of Massachusetts (US) 2008-07-02 EP disclosed
WO-2007002173-A1 HIV-1 PROTEASE INHIBITORS, AND METHODS OF MAKING AND USING THEM UNIVERSITY OF MASSACHUSETTS (US) 2007-01-04 WO disclosed