SCHEMBL4639384

SCHEMBL4639384

OC(C#Cc1ccccc1F)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 2/20 0.37
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
POLB P06746 3/20 0.35
TSHR P16473 1/20 0.34
PTGER4 P35408 2/20 0.34
GRM5 P41594 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C2 P52895 1/20 0.32
CYP19A1 P11511 1/20 0.32
RORC P51449 1/20 0.32
CETP P11597 1/20 0.32
CDC7 O00311 1/20 0.32
HSP90AA1 P07900 1/20 0.31
HSP90AB1 P08238 1/20 0.31
TACR1 P25103 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4639416 0.90 GRM2 (0.39) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4637798 0.88 ALDH1A1 (0.39) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4637803 0.86 CDC7 (0.37) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4638500 0.85 POLB (0.41) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4638930 0.84 ALDH1A1 (0.38) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4637824 0.80 ALDH1A1 (0.44) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4638086 0.78 TACR1 (0.39) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4637992 0.77 GRM2 (0.37) GRM2POLBPTGER4GRM5AKR1C3
SCHEMBL4637719 0.74 GRM2 (0.39) GRM2ALDH1A1GAAPOLBTSHR
SCHEMBL4637820 0.72 GAA (0.40) GRM2ALDH1A1GAAPOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed