SCHEMBL4637803

SCHEMBL4637803

OC(C#Cc1ccc(F)cc1)c1nnn(Cc2cc(C(F)(F)F)cc(C(F)(F)F)c2)c1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDC7 O00311 3/20 0.37
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
IDO1 P14902 1/20 0.35
TDO2 P48775 1/20 0.35
GRM2 Q14416 2/20 0.35
DAPK3 O43293 2/20 0.35
ROCK2 O75116 2/20 0.35
PRKD3 O94806 2/20 0.35
MAP4K4 O95819 2/20 0.35
PRKACA P17612 2/20 0.35
CDK2 P24941 2/20 0.35
FLT3 P36888 2/20 0.35
CLK2 P49760 2/20 0.35
GSK3B P49841 2/20 0.35
CDK9 P50750 2/20 0.35
PRKX P51817 2/20 0.35
JAK3 P52333 2/20 0.35
CDK5 Q00535 2/20 0.35
MAP4K2 Q12851 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637798 0.94 ALDH1A1 (0.39) ALDH1A1GAAGRM2POLBADORA3
SCHEMBL4638500 0.89 POLB (0.41) ALDH1A1GAAGRM2POLBADORA3
SCHEMBL4639384 0.86 GRM2 (0.37) CDC7ALDH1A1GAAGRM2POLB
SCHEMBL4638930 0.84 ALDH1A1 (0.38) ALDH1A1GAAGRM2POLBADORA3
SCHEMBL4639416 0.84 GRM2 (0.39) ALDH1A1GAAGRM2POLBADORA3
SCHEMBL4638482 0.80 ALDH1A1 (0.44) CDC7ALDH1A1GAAGRM2POLB
SCHEMBL4638086 0.78 TACR1 (0.39) ALDH1A1GAAGRM2POLBTSHR
SCHEMBL4638478 0.74 ADORA3 (0.41) CDC7ALDH1A1GAAIDO1TDO2
SCHEMBL4637719 0.74 GRM2 (0.39) ALDH1A1GAAGRM2POLBADORA3
SCHEMBL4637826 0.73 ALDH1A1 (0.47) ALDH1A1GAAGRM2POLBADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed