SCHEMBL4639434

SCHEMBL4639434

CON(C)C(=O)c1nnn(Cc2cc(Cl)cc(Cl)c2)c1-c1cccnc1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.42
P2RX7 Q99572 4/20 0.39
ALDH1A1 P00352 2/20 0.38
TSHR P16473 1/20 0.38
IDH1 O75874 1/20 0.36
KDR P35968 1/20 0.36
TEK Q02763 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NR1I3 Q14994 1/20 0.36
SLC16A3 O15427 1/20 0.35
CYP1A2 P05177 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HCRTR1 O43613 1/20 0.35
HCRTR2 O43614 1/20 0.35
HTR1A P08908 1/20 0.35
OPRM1 P35372 1/20 0.35
DRD3 P35462 1/20 0.35
HTR2B P41595 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4638522 0.88 CYP19A1 (0.44) CYP19A1P2RX7ALDH1A1TSHRNR1I3
SCHEMBL4637975 0.87 CYP19A1 (0.39) CYP19A1P2RX7ALDH1A1TSHRIDH1
SCHEMBL4637971 0.86 CYP19A1 (0.50) CYP19A1P2RX7ALDH1A1TSHRIDH1
SCHEMBL4637771 0.86 IDH1 (0.42) CYP19A1ALDH1A1IDH1KDRHCRTR1
SCHEMBL4638983 0.86 IDH1 (0.49) CYP19A1ALDH1A1TSHRIDH1
SCHEMBL4638860 0.84 CYP19A1 (0.46) CYP19A1P2RX7ALDH1A1TSHRIDH1
SCHEMBL4639523 0.83 MAPT (0.46) CYP19A1ALDH1A1IDH1L3MBTL1SMN1; SMN2
SCHEMBL4637939 0.78 POLQ (0.42) ALDH1A1IDH1KDR
SCHEMBL4638893 0.76 ABL1 (0.44) ALDH1A1KDRSMN1; SMN2HCRTR1HCRTR2
SCHEMBL4638811 0.75 IDH1 (0.40) CYP19A1P2RX7ALDH1A1TSHRIDH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed