SCHEMBL4638860

SCHEMBL4638860

O=C(O)c1nnn(Cc2cc(Cl)cc(Cl)c2)c1-c1cccnc1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 6/20 0.46
ALDH1A1 P00352 2/20 0.46
TSHR P16473 1/20 0.46
P2RX7 Q99572 4/20 0.45
HPGD P15428 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
MARS1 P56192 2/20 0.41
IDH1 O75874 1/20 0.40
HSD11B1 P28845 1/20 0.40
CYP2E1 P05181 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2A6 P11509 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2B6 P20813 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDR P35968 1/20 0.39
TEK Q02763 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637971 0.87 CYP19A1 (0.50) CYP19A1ALDH1A1TSHRP2RX7IDH1
SCHEMBL4639451 0.86 CYP19A1 (0.48) CYP19A1ALDH1A1TSHRP2RX7HPGD
SCHEMBL4637702 0.84 PTGER4 (0.44) CYP19A1ALDH1A1TSHRP2RX7HPGD
SCHEMBL4639434 0.84 CYP19A1 (0.42) CYP19A1ALDH1A1TSHRP2RX7L3MBTL1
SCHEMBL4637742 0.84 ALDH1A1 (0.52) CYP19A1ALDH1A1TSHRP2RX7HPGD
SCHEMBL4638551 0.83 IDH1 (0.55) CYP19A1ALDH1A1TSHRP2RX7HPGD
SCHEMBL4638811 0.81 IDH1 (0.40) CYP19A1ALDH1A1TSHRP2RX7L3MBTL1
SCHEMBL4638668 0.80 POLB (0.51) CYP19A1ALDH1A1P2RX7L3MBTL1IDH1
SCHEMBL4707264 0.75 RORB (0.49) ALDH1A1P2RX7L3MBTL1IDH1CYP2E1
SCHEMBL4638808 0.75 P2RX7 (0.38) ALDH1A1P2RX7L3MBTL1IDH1HSD11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501808-B1 TACHYKININ RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-07-02 EP disclosed