SCHEMBL4640645

SCHEMBL4640645

O=c1oc2c(I)c(O)ccc2c(Cc2ccc(OCCC3CCCN3)cc2)c1-c1ccc(Cl)cc1Cl

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 1/20 0.39
HSP90AB1 P08238 1/20 0.39
LTA4H P09960 5/20 0.37
AURKB Q96GD4 1/20 0.36
ESR1 P03372 2/20 0.35
PRKAB2 O43741 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA2 P54646 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAG3 Q9UGI9 1/20 0.35
PRKAG2 Q9UGJ0 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
SSTR2 P30874 2/20 0.33
CYP19A1 P11511 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5983904 0.87 ESR1 (0.48) LTA4HESR1CYP19A1
SCHEMBL4639644 0.87 LTA4H (0.45) HSP90AA1HSP90AB1LTA4HAURKBESR1
SCHEMBL4640758 0.85 LTA4H (0.46) LTA4HESR1
SCHEMBL4640684 0.84 ESR1 (0.38) ESR1CYP19A1
SCHEMBL6153596 0.84 CYP19A1 (0.51) LTA4HESR1CYP19A1
SCHEMBL6158194 0.78 ESR1 (0.45) ESR1
SCHEMBL6152270 0.78 ESR1 (0.47) ESR1
SCHEMBL5623982 0.76 LTA4H (0.46) LTA4HESR1
SCHEMBL5627051 0.75 LTA4H (0.44) LTA4HESR1
SCHEMBL6152455 0.75 CYP19A1 (0.44) ESR1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667999-A4 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARM LLC (US) 2008-08-06 EP disclosed
EP-1667999-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH Signal Pharmaceuticals LLC (US) 2006-06-14 EP disclosed
WO-2005028472-A1 BENZOPYRANONE COMPOUNDS, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2005-03-31 WO disclosed