SCHEMBL4640954

SCHEMBL4640954

N=C(N)NC1CCC(Nc2ncnc3c2ncn3CC(NC(=O)OCc2ccccc2)C(=O)O)CC1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.46
ITGAV P06756 10/20 0.46
TSHR P16473 1/20 0.42
ADORA1 P30542 2/20 0.42
HRH1 P35367 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
ITGA2B P08514 1/20 0.38
ITGB5 P18084 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4640963 1.00 ITGB3 (0.46) ITGB3ITGAVTSHRADORA1HRH1
SCHEMBL4640279 0.91 ITGB3 (0.48) ITGB3ITGAVADORA1HRH1
SCHEMBL4640271 0.91 ITGB3 (0.48) ITGB3ITGAVADORA1HRH1
SCHEMBL6810232 0.88 ITGB3 (0.46) ITGB3ITGAVTSHRADORA1
SCHEMBL6810237 0.88 ITGB3 (0.46) ITGB3ITGAVTSHRADORA1
SCHEMBL6805719 0.83 BTK (0.42) ITGB3ITGAVADORA1
SCHEMBL4644200 0.83 BTK (0.42) ITGB3ITGAVADORA1
SCHEMBL6911764 0.83 ADORA1 (0.40) ITGB3ITGAVTSHRADORA1CNR1
SCHEMBL4641275 0.81 ITGB3 (0.43) ITGB3ITGAVADORA1
SCHEMBL4641283 0.81 ITGB3 (0.46) ITGB3ITGAVADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed