SCHEMBL4640975

SCHEMBL4640975

c1ccc(C2=NOC3(CCCCCC(c4ccccc4)CC3)C2)cc1

nearest known ligand 0.49

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRNB4 P30926 1/20 0.49
CHRNA3 P32297 1/20 0.49
CYP2C9 P11712 8/20 0.36
KCNH2 Q12809 1/20 0.36
TRPM8 Q7Z2W7 1/20 0.36
SLC18A3 Q16572 2/20 0.35
POLB P06746 1/20 0.35
CASP3 P42574 1/20 0.35
SENP7 Q9BQF6 1/20 0.35
SENP6 Q9GZR1 1/20 0.35
HTR1A P08908 1/20 0.34
ADRA1B P35368 1/20 0.34
CCR5 P51681 2/20 0.34
CYP11B2 P19099 1/20 0.34
TRPA1 O75762 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2210855 0.92 CHRNB4 (0.49) CHRNB4CHRNA3SLC18A3POLB
SCHEMBL4639958 0.92 CHRNB4 (0.45) CHRNB4CHRNA3CYP2C9KCNH2TRPM8
SCHEMBL4640229 0.89 CHRNB4 (0.42) CHRNB4CHRNA3CYP2C9KCNH2TRPM8
SCHEMBL4639854 0.89 CYP2C9 (0.41) CHRNB4CHRNA3CYP2C9KCNH2TRPM8
SCHEMBL4640438 0.84 NPC1 (0.39) CHRNB4CHRNA3CYP2C9KCNH2TRPM8
SCHEMBL4620189 0.83 NLRP3 (0.47) CHRNB4CHRNA3POLB
SCHEMBL2208302 0.80 CHRNB4 (0.42) CHRNB4CHRNA3CYP2C9
SCHEMBL4621179 0.75 SCD5 (0.39) CHRNB4CHRNA3CYP2C9SLC18A3POLB
SCHEMBL5011255 0.75 KMT2A (0.43) CHRNB4CHRNA3POLB
SCHEMBL2207499 0.75 CHRNB4 (0.49) CHRNB4CHRNA3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO claimed