SCHEMBL4640438

SCHEMBL4640438

c1ccc(C2CCCCCC3(CC2)CC(c2ccccn2)=NO3)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.39
MAPK1 P28482 2/20 0.39
RAB9A P51151 2/20 0.39
ALDH1A1 P00352 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
TP53 P04637 1/20 0.39
SCD5 Q86SK9 3/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
HSD17B10 Q99714 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
SCD O00767 1/20 0.34
CYP11B2 P19099 1/20 0.33
HSP90AA1 P07900 1/20 0.33
SLC2A1 P11166 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
NCOA1 Q15788 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4621179 0.93 SCD5 (0.39) NPC1MAPK1RAB9AALDH1A1SMN1; SMN2
SCHEMBL4640975 0.84 CHRNB4 (0.49) CHRNB4CHRNA3CYP11B2SLC18A3CCR5
SCHEMBL4639958 0.80 CHRNB4 (0.45) NPC1RAB9AALDH1A1CHRNB4CHRNA3
SCHEMBL4643609 0.78 NPC1 (0.34) NPC1MAPK1RAB9AALDH1A1SMN1; SMN2
SCHEMBL4640229 0.77 CHRNB4 (0.42) TP53CHRNB4CHRNA3S1PR1SLC18A3
SCHEMBL4639854 0.77 CYP2C9 (0.41) ALDH1A1KDM4EHSD17B10CHRNB4CHRNA3
SCHEMBL2210855 0.76 CHRNB4 (0.49) ALDH1A1KDM4ECHRNB4CHRNA3SLC18A3
SCHEMBL2209482 0.71 GAA (0.35) NPC1MAPK1RAB9ASMN1; SMN2KDM4E
SCHEMBL4620189 0.71 NLRP3 (0.47) NPC1RAB9AALDH1A1SMN1; SMN2CHRNB4
SCHEMBL12901458 0.69 SLC18A3 (0.37) ALDH1A1SLC18A3HTR1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO claimed