SCHEMBL4641010

SCHEMBL4641010

O=C(N[C@@H](Cn1cnc2c(NCCCCNc3nc4ccccc4[nH]3)ncnc21)C(=O)O)OCc1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 19/20 0.68
ITGAV P06756 19/20 0.68
ITGA2B P08514 2/20 0.53
ITGB5 P18084 2/20 0.53
HDAC1 Q13547 1/20 0.46
HDAC2 Q92769 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641327 0.92 ITGB3 (0.59) ITGB3ITGAVITGA2BITGB5HDAC1
SCHEMBL6805087 0.84 ITGB3 (0.57) ITGB3ITGAVITGA2BITGB5HDAC1
SCHEMBL6806785 0.80 ITGB3 (0.51) ITGB3ITGAVITGA2BITGB5HDAC1
SCHEMBL4640796 0.77 ITGB3 (0.47) ITGB3ITGAVHDAC1HDAC2
SCHEMBL4640793 0.77 ITGB3 (0.47) ITGB3ITGAVHDAC1HDAC2
SCHEMBL6806782 0.76 ITGB3 (0.46) ITGB3ITGAVITGA2BITGB5HDAC1
SCHEMBL5840142 0.76 HDAC6 (0.47) ITGB3ITGAV
SCHEMBL4641275 0.74 ITGB3 (0.43) ITGB3ITGAVHDAC1HDAC2
SCHEMBL4641283 0.74 ITGB3 (0.46) ITGB3ITGAVHDAC1HDAC2
SCHEMBL6804197 0.73 ITGB3 (0.47) ITGB3ITGAVHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0853084-B1 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AG (DE) 2008-08-13 EP disclosed
US-6723727-B1 VITRONECTIN RECEPTOR ANTAGONISTS; INHIBITORS OF BONE RESORPTION; OSTEOPOROSIS HOECHST AKTIENGESELLSCHAFT (DE) 2004-04-20 US disclosed
EP-0853084-A2 Substituted purine derivatives as vitronectin receptor antagonists HOECHST AKTIENGESELLSCHAFT (DE) 1998-07-15 EP disclosed