SCHEMBL4642121

SCHEMBL4642121

Cc1cccc(C#Cc2cc3c(c(C(=O)O)c2)OC(C)(C)C=C3)c1C(N)=O

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
PTPN1 P18031 1/20 0.32
FFAR1 O14842 1/20 0.31
IKBKB O14920 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4641330 0.74 HDAC8 (0.35)
SCHEMBL4961626 0.70 ALDH1A1 (0.33)
SCHEMBL8940635 0.63 NPC1 (0.68) NPC1RAB9AFFAR1
SCHEMBL11245121 0.62 ALDH1A1 (0.57) NPC1RAB9A
SCHEMBL13805579 0.60 HTR2C (0.55) NPC1RAB9APTPN1
SCHEMBL30937310 0.60 ALDH1A1 (0.50) PTPN1
SCHEMBL4641291 0.59 COXFA4 (0.44)
SCHEMBL6029391 0.59 ALDH1A1 (0.52) NPC1RAB9A
SCHEMBL2540273 0.58 PARP1 (0.46)
SCHEMBL311565 0.58 PARP1 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1956016-A1 Bicyclic acyltryptophanols Bayer Schering Pharma Aktiengesellschaft (DE) 2008-08-13 EP disclosed