SCHEMBL4643609

SCHEMBL4643609

CCC(C)(C)C1CCCCCC2(CC1)CC(c1ccccn1)=NO2

nearest known ligand 0.34

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.34
RAB9A P51151 2/20 0.34
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TP53 P04637 1/20 0.32
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CYP2C9 P11712 9/20 0.31
KCNH2 Q12809 1/20 0.31
TRPM8 Q7Z2W7 1/20 0.31
MAPT P10636 1/20 0.30
S1PR1 P21453 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2209482 0.94 GAA (0.35) NPC1RAB9AKDM4EGAACHRNB4
SCHEMBL4640438 0.78 NPC1 (0.39) NPC1RAB9AKDM4ECHRNB4CHRNA3
SCHEMBL4621179 0.72 SCD5 (0.39) NPC1RAB9AKDM4ECHRNB4CHRNA3
SCHEMBL2206353 0.71 CHRNB4 (0.34) NPC1RAB9AKDM4EGAACHRNB4
SCHEMBL10210782 0.68 CHRNB4 (0.38) KDM4ECHRNB4CHRNA3ALDH1A1MAPK1
SCHEMBL10168567 0.65 CHRNB4 (0.36) CHRNB4CHRNA3MAPK1CYP2C9
SCHEMBL2205238 0.64 KDM4E (0.37) KDM4EGAAALDH1A1MAPT
SCHEMBL17300431 0.64 NPC1 (0.39) NPC1KDM4EALDH1A1SMN1; SMN2CYP2C9
SCHEMBL4641139 0.64 CHRNB4 (0.37) GAACHRNB4CHRNA3ALDH1A1TP53
SCHEMBL4640975 0.62 CHRNB4 (0.49) CHRNB4CHRNA3CYP2C9KCNH2TRPM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888542-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006136245-A1 SUBSTITUTED SPIRO-COMPOUNDS AND THE USE THEREOF FOR PRODUCING MEDICAMENTS Grünenthal GmbH (DE) 2006-12-28 WO claimed