SCHEMBL4644282

SCHEMBL4644282

Cc1cc(C)nc(N(c2ccccc2)C(Oc2cccc3[nH]c4ccccc4c23)C(C)O)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.40
DNM1 Q05193 2/20 0.40
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
HTT P42858 1/20 0.39
TLR4 O00206 6/20 0.37
GABRP O00591 1/20 0.35
GABRD O14764 1/20 0.35
GABRA1 P14867 1/20 0.35
GABRB1 P18505 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
GABRB2 P47870 1/20 0.35
GABRA4 P48169 1/20 0.35
GABRE P78334 1/20 0.35
GABRA6 Q16445 1/20 0.35
GABRG1 Q8N1C3 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4605327 0.75 ADRB2 (0.45) ADRB2DNM1KDM4ELMNAHTT
SCHEMBL4644273 0.74 TLR4 (0.53) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4608624 0.72 ADRB2 (0.47) ADRB2DNM1KDM4ETLR4ADRB3
SCHEMBL4606845 0.68 ADRB2 (0.42) ADRB2DNM1KDM4ETLR4GABRP
SCHEMBL1733165 0.68 KMT2A (0.54) ADRB2DNM1LMNATLR4GABRP
SCHEMBL4608341 0.67 ADRB2 (0.53) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4436284 0.67 ADRB2 (0.55) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL9621537 0.67 ADRB2 (0.55) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4605235 0.66 TUBB4A (0.48) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4779938 0.66 ADRB2 (0.51) ADRB2DNM1KDM4ELMNATLR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP disclosed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO disclosed