SCHEMBL4605327

SCHEMBL4605327

Cc1cc(C)nc(NC(Oc2cccc3[nH]c4ccccc4c23)C(C)O)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 7/20 0.45
DNM1 Q05193 2/20 0.45
KDM4E B2RXH2 2/20 0.41
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
TLR4 O00206 5/20 0.41
ADRB3 P13945 2/20 0.39
DRD2 P14416 3/20 0.38
MAPT P10636 2/20 0.38
SLC22A2 O15244 1/20 0.38
SLC22A1 O15245 1/20 0.38
MLNR O43193 1/20 0.38
NR1I2 O75469 1/20 0.38
KCNK2 O95069 1/20 0.38
ABCB11 O95342 1/20 0.38
APP P05067 1/20 0.38
ABCB1 P08183 1/20 0.38
ADRB1 P08588 1/20 0.38
HTR1A P08908 1/20 0.38
ADRA2A P08913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4608341 0.80 ADRB2 (0.53) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL9621537 0.79 ADRB2 (0.55) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4727264 0.77 ADRB2 (0.50) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4607220 0.75 ADRB3 (0.48) ADRB2DNM1KDM4ETLR4ADRB3
SCHEMBL6507182 0.75 ADRB2 (0.54) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4644282 0.75 ADRB2 (0.40) ADRB2DNM1KDM4ELMNAHTT
SCHEMBL2992618 0.74 TLR4 (0.67) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4457452 0.74 ADRB2 (0.53) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4795725 0.73 ADRB2 (0.49) ADRB2DNM1KDM4ELMNATLR4
SCHEMBL4643608 0.72 ADRB3 (0.46) ADRB2DNM1KDM4ETLR4ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1945612-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS Orchid Research Laboratories Limited (IN) 2008-07-23 EP claimed
WO-2007042912-A2 HETEROCYCLIC COMPOUNDS AS PSTAT3/IL-6 INHIBITORS ORCHID RESEARCH LABORATORIES LIMITED (IN) 2007-04-19 WO claimed