SCHEMBL4645586

SCHEMBL4645586

COc1ccc([C@@H](C(=O)O)C2(O)CCCCC2I)cc1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 4/20 0.39
SLC6A4 P31645 4/20 0.39
SLC6A3 Q01959 4/20 0.39
LMNA P02545 1/20 0.39
CNR1 P21554 1/20 0.39
HTR2A P28223 1/20 0.39
HRH1 P35367 1/20 0.39
HRH3 Q9Y5N1 1/20 0.39
ALDH1A1 P00352 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
MAPK1 P28482 1/20 0.38
CYP2C19 P33261 1/20 0.38
MMP1 P03956 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP13 P45452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4643005 0.79 ITGA4 (0.40) ALDH1A1
SCHEMBL13637842 0.77 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3LMNACNR1
SCHEMBL4510516 0.77 SLC6A2 (0.55) SLC6A2SLC6A4SLC6A3LMNACNR1
SCHEMBL11834256 0.71 GAA (0.39) SLC6A4SLC6A3LMNAALDH1A1MAPK1
SCHEMBL17296892 0.70 ATM (0.47) SLC6A2SLC6A4SLC6A3LMNACNR1
SCHEMBL7704043 0.69 SLC6A4 (0.45) SLC6A2SLC6A4SLC6A3LMNACNR1
SCHEMBL1566474 0.68 ALOX5 (0.51) SLC6A2SLC6A4SLC6A3ALDH1A1MMP1
SCHEMBL11848170 0.68 MME (0.40) SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL10616814 0.67 SLC6A2 (0.56) SLC6A2SLC6A4SLC6A3LMNACNR1
SCHEMBL3952145 0.67 SLC6A2 (0.46) SLC6A2SLC6A4SLC6A3LMNACNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1957470-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS Wyeth (US) 2008-08-20 EP disclosed
WO-2007067501-A1 PROCESS FOR SELECTIVE SYNTHESIS OF ENANTIOMERS OF SUBSTITUTED 1-(2-AMINO-1-PHENYL-ETHYL)-CYCLOHEXANOLS WYETH (US) 2007-06-14 WO disclosed