SCHEMBL4647436

SCHEMBL4647436

O=CCc1cc(F)ccc1[N+](=O)[O-]

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
SNCA P37840 4/20 0.44
ALDH1A1 P00352 8/20 0.43
MAPT P10636 3/20 0.43
MAPK1 P28482 1/20 0.43
HSPB1 P04792 3/20 0.39
HTT P42858 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PDE7A Q13946 1/20 0.38
POLB P06746 1/20 0.38
KDM4E B2RXH2 1/20 0.37
KMT2A Q03164 1/20 0.37
TSHR P16473 1/20 0.37
HIF1A Q16665 1/20 0.37
KCNMA1 Q12791 1/20 0.37
ALDH3A1 P30838 1/20 0.36
RIPK1 Q13546 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL621196 0.86 TDP1 (0.50) ATMTDP1SNCAALDH1A1MAPT
SCHEMBL310240 0.85 ATM (0.53) ATMTDP1SNCAALDH1A1MAPT
SCHEMBL29362511 0.80 TDP1 (0.60) ATMTDP1SNCAALDH1A1MAPT
SCHEMBL310839 0.80 TDP1 (0.60) ATMTDP1SNCAALDH1A1MAPT
SCHEMBL405343 0.79 ACHE (0.40) ATMTDP1ALDH1A1MAPK1KMT2A
SCHEMBL405093 0.79 TSHR (0.55) ATMALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL406455 0.79 TSHR (0.56) ALDH1A1MAPTKMT2ATSHR
SCHEMBL12246128 0.79 ALDH1A1 (0.44) TDP1ALDH1A1MAPTMAPK1SMN1; SMN2
SCHEMBL463502 0.79 TSHR (0.36) ATMTDP1ALDH1A1MAPTMAPK1
SCHEMBL2891144 0.79 TDP1 (0.58) ATMTDP1SNCAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1667989-A4 SUBSTITUTED ISOQUINOLINONES PORTOLA PHARM INC (US) 2008-08-20 EP disclosed
EP-1667989-A1 SUBSTITUTED ISOQUINOLINONES Portola Pharmaceuticals, Inc. (US) 2006-06-14 EP disclosed
WO-2005035520-A1 SUBSTITUTED ISOQUINOLINONES PORTOLA PHARMACEUTICALS, INC. (US) 2005-04-21 WO disclosed