SCHEMBL464765

SCHEMBL464765

CCOC(=O)C1CC(O)CN1C

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.37
MEN1 O00255 2/20 0.37
ATM Q13315 1/20 0.37
MAPT P10636 3/20 0.36
ALDH1A1 P00352 7/20 0.36
LMNA P02545 1/20 0.36
FKBP1A P62942 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL464766 1.00 KMT2A (0.37) KMT2AMEN1ATMMAPTALDH1A1
SCHEMBL20113215 1.00 KMT2A (0.37) KMT2AMEN1ATMMAPTALDH1A1
SCHEMBL4886758 0.81 POLB (0.43) KMT2AMEN1ATMALDH1A1LMNA
SCHEMBL4886754 0.81 POLB (0.43) KMT2AMEN1ATMALDH1A1LMNA
SCHEMBL7306693 0.81 KMT2A (0.36) KMT2AMEN1ATMMAPTALDH1A1
SCHEMBL7302241 0.81 KMT2A (0.36) KMT2AMEN1ATMMAPTALDH1A1
SCHEMBL26078627 0.81 KMT2A (0.36) KMT2AMEN1MAPTALDH1A1LMNA
SCHEMBL14288714 0.81 MMP2 (0.42) KMT2AMEN1MAPTALDH1A1LMNA
SCHEMBL7308325 0.81 KMT2A (0.36) KMT2AMEN1ATMMAPTALDH1A1
SCHEMBL16367126 0.81 KMT2A (0.36) KMT2AMEN1ATMMAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080176923-A1 Proline Derivatives Used as Pharmaceutical Active Ingredients for the Treatment of Tumors SALAMA ZOSER B 2008-07-24 US claimed
WO-2022078462-A1 NOVEL GLUTAMINE ANALOGS JACOBIO PHARMACEUTICALS CO., LTD. (CN) 2022-04-21 WO disclosed
EP-1765328-B1 ANTI-CANCER COMPOSITION COMPRISING PROLINE OR ITS DERIVATIVES AND AN ANTI-TUMOUR ANTIBODY SALAMA ZOSER B (DE) 2011-11-23 EP disclosed
US-7727530-B2 Anti-cancer composition comprising proline or its derivatives and an anti-tumour antibody SALAMA ZOSER B 2010-06-01 US disclosed
US-20080176923-A1 Proline Derivatives Used as Pharmaceutical Active Ingredients for the Treatment of Tumors SALAMA ZOSER B 2008-07-24 US disclosed
US-20080176923-A1 Proline Derivatives Used as Pharmaceutical Active Ingredients for the Treatment of Tumors SALAMA ZOSER B 2008-07-24 US disclosed
US-20050276810-A1 Anti-cancer composition comprising proline or its derivatives and an anti-tumour antibody SALAMA ZOSER B 2005-12-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080176923-A1 Proline Derivatives Used as Pharmaceutical Active Ingredients for the Treatment of Tumors PREP, PRAP1, VHL KMT2A 2637/4885MEN1 660/4885ATM 3665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.