N,N-Dimethylethanaminium

N,N-Dimethylethanaminium

SCHEMBL4648022

CCC=C(C)C(=O)OCC.CCN(C)C.O=S(=O)(O)O

nearest known ligand 0.38

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of N,N-Dimethylethanaminium. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GLO1 Q04760 1/20 0.38
CYP2D6 P10635 2/20 0.38
CYP2C19 P33261 1/20 0.38
CYP2C9 P11712 1/20 0.36
NPSR1 Q6W5P4 2/20 0.34
ALDH1A1 P00352 5/20 0.33
LMNA P02545 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MAPT P10636 2/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
S1PR4 O95977 1/20 0.31
S1PR1 P21453 1/20 0.31
MAPK1 P28482 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TRPA1 O75762 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfuric Acid SCHEMBL3054230 0.93 GLO1 (0.40) GLO1CYP2D6CYP2C19CYP2C9NPSR1
Trimethylammonium SCHEMBL17712424 0.86 GLO1 (0.45) GLO1CYP2D6CYP2C19CYP2C9NPSR1
Trimethylammonium SCHEMBL16429829 0.86 GLO1 (0.45) GLO1CYP2D6CYP2C19CYP2C9NPSR1
SCHEMBL134789 0.84 GLO1 (0.50) GLO1CYP2D6CYP2C19CYP2C9NPSR1
SCHEMBL1618911 0.84 GLO1 (0.50) GLO1CYP2D6CYP2C19CYP2C9NPSR1
Sulfuric Acid SCHEMBL16660529 0.82 CHRM1 (0.42) CYP2C19NPSR1ALDH1A1LMNAMAPT
Sulfuric Acid SCHEMBL28116564 0.82 CHRM1 (0.42) CYP2C19NPSR1ALDH1A1LMNAMAPT
Water SCHEMBL7175634 0.82 GLO1 (0.48) GLO1CYP2D6CYP2C19CYP2C9NPSR1
Sulfuric Acid SCHEMBL2378917 0.79 GLO1 (0.42) GLO1CYP2D6CYP2C19CYP2C9NPSR1
Dimethylamine SCHEMBL447225 0.78 GLO1 (0.45) GLO1CYP2D6CYP2C19CYP2C9NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1687348-B1 COPOLYMERS COMPRISING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS BASF SE (DE) 2008-11-12 EP claimed
EP-3467086-B1 DISHWASHING CLEANING COMPOSITION PROCTER & GAMBLE (US) 2021-03-24 EP disclosed
US-10815327-B2 Copolymers comprising polyalkylene oxide groups and quaternary nitrogen atoms BASF SE (DE) 2020-10-27 US disclosed
US-10731106-B2 Dishwashing cleaning composition THE PROCTER & GAMBLE COMPANY (US) 2020-08-04 US disclosed
US-10723979-B2 Dishwashing cleaning composition THE PROCTER & GAMBLE COMPANY (US) 2020-07-28 US disclosed
EP-3440121-B1 COPOLYMERS COMPRISING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS BASF SE (DE) 2020-05-06 EP disclosed
EP-3228687-B1 DISHWASHING CLEANING COMPOSITION PROCTER & GAMBLE (US) 2019-05-22 EP disclosed
US-20190106658-A1 DISHWASHING CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY 2019-04-11 US disclosed
WO-2019070924-A1 DISHWASHING CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2019-04-11 WO disclosed
WO-2019070923-A1 DISHWASHING CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2019-04-11 WO disclosed
EP-3440121-A1 COPOLYMERS COMPRISING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS BASF SE (DE) 2019-02-13 EP disclosed
US-20170292093-A1 DISHWASHING CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY 2017-10-12 US disclosed
WO-2017174468-A1 COPOLYMERS COMPRISING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS BASF SE (DE) 2017-10-12 WO disclosed
WO-2017176500-A1 DISHWASHING CLEANING COMPOSITION THE PROCTER & GAMBLE COMPANY (US) 2017-10-12 WO disclosed
EP-3228687-A1 DISHWASHING CLEANING COMPOSITION The Procter and Gamble Company (US) 2017-10-11 EP disclosed
EP-1685227-B1 LAUNDRY COMPOSITIONS HAVING COPOLYMERS CONTAINING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS AND A SURFACTANT SYSTEM PROCTER & GAMBLE (US) 2008-08-20 EP disclosed
US-20070129516-A1 Copolymers comprising polyalkylene oxide groups and quaternary nitrogen atoms DETERING JUERGEN 2007-06-07 US disclosed
EP-1685227-A1 LAUNDRY COMPOSITIONS HAVING COPOLYMERS CONTAINING POLYALKYLENE OXIDE GROUPS AND QUATERNARY NITROGEN ATOMS AND A SURFACTANT SYSTEM THE PROCTER & GAMBLE COMPANY (US) 2006-08-02 EP disclosed
WO-2005052107-A1 LAUNDRY COMPOSITIONS HAVING COPOLYMERS CONTAINING POLYALKYLENE OXIDE GROUPS AND QUANTERNARY NITROGEN ATOMS AND A SURFACTANT SYSTEM THE PROCTER & GAMBLE COMPANY (US) 2005-06-09 WO disclosed
US-20050113280-A1 Laundry compositions having copolymers containing polyalkylene oxide groups and quaternary nitrogen atoms and a surfactant system PROCTER & GAMBLE COMPANY, THE 2005-05-26 US disclosed