SCHEMBL4649642

SCHEMBL4649642

NC1CCC(NS(=O)(=O)c2ccc(CNc3nccc(Nc4ccc(F)cc4)n3)cc2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 10/20 0.46
CA1 P00915 8/20 0.46
MEN1 O00255 1/20 0.45
NPC1 O15118 1/20 0.45
LMNA P02545 1/20 0.45
MAPT P10636 1/20 0.45
ALOX12 P18054 1/20 0.45
MAPK1 P28482 1/20 0.45
RAB9A P51151 1/20 0.45
KMT2A Q03164 1/20 0.45
NAMPT P43490 2/20 0.44
ACHE P22303 1/20 0.41
BACE1 P56817 1/20 0.41
CCNA2 P20248 2/20 0.41
CDK2 P24941 2/20 0.41
CCNE2 O96020 1/20 0.41
CCNE1 P24864 1/20 0.41
CCNA1 P78396 1/20 0.41
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4687574 0.86 ACHE (0.49) CA2CA1MEN1NPC1LMNA
SCHEMBL4909568 0.81 ACHE (0.48) CA2MEN1NPC1LMNAMAPT
SCHEMBL4623805 0.74 HTR7 (0.49) CA2CA1MEN1NPC1LMNA
SCHEMBL13392500 0.73 MAPT (0.56) CA2CA1MEN1NPC1LMNA
Hydrochloric Acid SCHEMBL4904480 0.73 NAMPT (0.41) CA2CA1NAMPTCDK2CCNE1
SCHEMBL4649640 0.72 MEN1 (0.53) CA2CA1MEN1NPC1LMNA
SCHEMBL3298093 0.72 MAPT (0.50) MEN1NPC1LMNAMAPTALOX12
SCHEMBL4623995 0.72 HTR1A (0.47) CA2CA1MEN1NPC1LMNA
Hydrochloric Acid SCHEMBL4881165 0.72 MEN1 (0.52) CA2CA1MEN1NPC1LMNA
SCHEMBL4653131 0.70 MEN1 (0.61) CA2CA1MEN1NPC1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904479-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS Sanofi-Aventis (FR) 2008-04-02 EP disclosed
WO-2007006926-A2 NOVEL 2,4-DIANILINOPYRIMIDINE DERIVATIVES, THE PREPARATION THEREOF, THEIR USE AS MEDICAMENTS, PHARMACEUTICAL COMPOSITIONS AND, IN PARTICULAR, AS IKK INHIBITORS SANOFI-AVENTIS (FR) 2007-01-18 WO disclosed