SCHEMBL4649736

SCHEMBL4649736

CC(C)c1cc(Nc2ccc(F)cc2F)ncc1CN(C)C1CCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 1/20 0.38
CDK2 P24941 1/20 0.38
EGFR P00533 1/20 0.35
GAA P10253 2/20 0.34
POLB P06746 1/20 0.34
PIK3CA P42336 1/20 0.34
PRKDC P78527 1/20 0.34
CNR2 P34972 3/20 0.34
SLC6A4 P31645 2/20 0.33
RECQL P46063 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A3 Q01959 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
ALDH1A1 P00352 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4649780 0.83 CNR2 (0.37) CNR2SLC6A4SLC6A2SLC6A3CYP3A4
SCHEMBL4649692 0.82 CNR2 (0.50) POLBCNR2CYP1A2CYP3A4CYP2D6
SCHEMBL4649737 0.81 CNR2 (0.42) CDK4CDK2GAAPOLBPIK3CA
SCHEMBL4649712 0.81 CNR2 (0.54) EGFRPIK3CACNR2SLC6A4SLC6A2
SCHEMBL4650258 0.80 CNR2 (0.33) CNR2
SCHEMBL4649624 0.80 CNR2 (0.42) CDK4CDK2POLBCNR2CYP1A2
SCHEMBL4649071 0.79 CNR2 (0.37) CDK4CNR2CYP1A2CYP2C9CYP2C19
SCHEMBL4649170 0.77 CNR2 (0.55) EGFRPIK3CACNR2SLC6A4SLC6A2
SCHEMBL4649775 0.76 CNR2 (0.40) POLBCNR2CYP1A2CYP3A4CYP2D6
SCHEMBL4649631 0.76 CNR2 (0.56) CDK2EGFRGAAPOLBPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1718613-B1 PYRIDINE DERIVATIVES AND THEIR USE AS CB2 RECEPTOR MODULATORS GLAXO GROUP LTD (GB) 2008-09-03 EP disclosed