SCHEMBL4649972

SCHEMBL4649972

Cc1cccc(CNC(=O)[C@H](CCC(=O)O)NC(=O)c2ccc(-c3ccc4c(c3)OCO4)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.52
TDP1 Q9NUW8 1/20 0.48
MMP2 P08253 1/20 0.48
ADAMTS4 O75173 1/20 0.47
ADAMTS5 Q9UNA0 1/20 0.47
CHRM3 P20309 4/20 0.46
P2RY12 Q9H244 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
USP2 O75604 1/20 0.46
LMNA P02545 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
CYP2C9 P11712 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
CYP2C19 P33261 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2247941 0.88 MMP2 (0.56) MMP2ADAMTS4ADAMTS5P2RY12CTSB
SCHEMBL2247356 0.83 MMP2 (0.57) HPGDTDP1MMP2ADAMTS4ADAMTS5
SCHEMBL3583743 0.79 ADAMTS5 (0.56) MMP2ADAMTS4ADAMTS5P2RY12CTSB
SCHEMBL3576509 0.78 ADAMTS5 (0.62) MMP2ADAMTS4ADAMTS5MAPK1CTSB
SCHEMBL2246985 0.77 ADAMTS5 (0.59) MMP2ADAMTS4ADAMTS5MEN1KMT2A
SCHEMBL2246335 0.77 MMP2 (0.58) MMP2ADAMTS4ADAMTS5CTSBCTSL
SCHEMBL3591190 0.77 CTSB (0.55) MMP2ADAMTS4ADAMTS5CTSBCTSL
SCHEMBL2245471 0.77 MMP2 (0.69) MMP2ADAMTS4ADAMTS5CTSBCTSL
SCHEMBL2244723 0.77 ADAMTS5 (0.56) MMP2ADAMTS4ADAMTS5CTSBCTSL
SCHEMBL2247357 0.76 MMP2 (0.61) MMP2ADAMTS4ADAMTS5CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1902014-A2 GLUTAMATE AGGRECANASE INHIBITORS Wyeth (US) 2008-03-26 EP disclosed
WO-2007008994-A2 GLUTAMATE AGGRECANASE INHIBITORS WYETH (US) 2007-01-18 WO disclosed