SCHEMBL4650682

SCHEMBL4650682

O=C(O)c1c[nH]c2c(F)cc(Cc3c(F)cccc3C(F)(F)F)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
RAB9A P51151 1/20 0.42
ALDH1A1 P00352 4/20 0.41
HPGD P15428 3/20 0.41
CYP1A2 P05177 2/20 0.41
MEN1 O00255 1/20 0.41
ALOX12 P18054 1/20 0.41
KMT2A Q03164 1/20 0.41
LMNA P02545 1/20 0.40
CSNK2A2 P19784 2/20 0.39
CSNK2B P67870 2/20 0.39
CSNK2A1 P68400 2/20 0.39
FABP4 P15090 1/20 0.39
DNA2 P51530 1/20 0.38
CASP6 P55212 1/20 0.38
CTDSP1 Q9GZU7 1/20 0.38
GUSB P08236 2/20 0.37
TET2 Q6N021 1/20 0.37
TET1 Q8NFU7 1/20 0.37
RORC P51449 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650046 0.90 RAB9A (0.47) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650636 0.87 KDM4E (0.43) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650015 0.86 ALDH1A1 (0.42) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4649260 0.83 RAB9A (0.42) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4649428 0.82 ALDH1A1 (0.45) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650022 0.82 ALDH1A1 (0.50) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4649447 0.81 RAB9A (0.49) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650802 0.81 ALDH1A1 (0.53) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650037 0.81 RAB9A (0.45) KDM4ERAB9AALDH1A1HPGDCYP1A2
SCHEMBL4650127 0.80 KDM4A (0.48) KDM4ERAB9AALDH1A1HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed