SCHEMBL4650127

SCHEMBL4650127

O=C(O)c1c[nH]c2c(F)cc(Cc3ccc(Cl)c(C(F)(F)F)c3)cc2c1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4A O75164 1/20 0.48
KDM5A P29375 1/20 0.48
KDM5B Q9UGL1 1/20 0.48
CSNK2A2 P19784 4/20 0.46
CSNK2B P67870 4/20 0.46
CSNK2A1 P68400 4/20 0.46
ALDH1A1 P00352 2/20 0.41
CYP1A2 P05177 2/20 0.41
MEN1 O00255 1/20 0.41
HPGD P15428 1/20 0.41
ALOX12 P18054 1/20 0.41
KMT2A Q03164 1/20 0.41
MDH2 P40926 1/20 0.40
LMNA P02545 1/20 0.40
KDM4E B2RXH2 2/20 0.38
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
ABCB11 O95342 1/20 0.36
NOTUM Q6P988 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4650045 0.85 ALDH1A1 (0.46) ALDH1A1CYP1A2MEN1HPGDALOX12
SCHEMBL4650041 0.85 ALDH1A1 (0.47) KDM5AKDM5BCSNK2A2CSNK2BCSNK2A1
SCHEMBL4650802 0.84 ALDH1A1 (0.53) KDM5AKDM5BCSNK2A2CSNK2BCSNK2A1
SCHEMBL4649455 0.83 ALDH1A1 (0.50) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4650022 0.81 ALDH1A1 (0.50) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4650015 0.81 ALDH1A1 (0.42) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4650682 0.80 KDM4E (0.43) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4649447 0.80 RAB9A (0.49) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4650793 0.80 ALDH1A1 (0.46) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2
SCHEMBL4650636 0.80 KDM4E (0.43) CSNK2A2CSNK2BCSNK2A1ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963271-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS Merck & Co., Inc. (US) 2008-09-03 EP claimed
WO-2007067489-A1 QUINOLONE M1 RECEPTOR POSITIVE ALLOSTERIC MODULATORS MERCK & CO., INC. (US) 2007-06-14 WO claimed