SCHEMBL4654495

SCHEMBL4654495

O=C1NCC(CCCC(c2ccc(F)cc2)c2ccc(F)cc2)N1CC=Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 5/20 0.44
KMT2A Q03164 5/20 0.44
MAPT P10636 5/20 0.44
LMNA P02545 5/20 0.44
CYP2D6 P10635 4/20 0.44
OPRM1 P35372 4/20 0.44
HIF1A Q16665 3/20 0.44
SLC6A4 P31645 3/20 0.44
SLC6A3 Q01959 3/20 0.44
CYP1A2 P05177 3/20 0.44
CYP3A4 P08684 3/20 0.44
CYP2C9 P11712 3/20 0.44
MAPK1 P28482 3/20 0.44
SIGMAR1 Q99720 2/20 0.44
THPO P40225 2/20 0.44
ADORA3 P0DMS8 2/20 0.44
DRD2 P14416 2/20 0.44
ADRA2B P18089 2/20 0.44
ADRA2C P18825 2/20 0.44
CHRM3 P20309 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4654585 0.78 CYP3A4 (0.46) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL4653378 0.77 MEN1 (0.46) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL4653345 0.75 MAPT (0.44) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL4653651 0.74 LMNA (0.44) MAPTLMNASIGMAR1NPSR1KDM4E
SCHEMBL4652287 0.73 CYP3A4 (0.41) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL4289774 0.73 MEN1 (0.51) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL4289771 0.73 MEN1 (0.51) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL28392280 0.64 LMNA (0.72) MEN1KMT2AMAPTLMNACYP2D6
Flunarizine SCHEMBL1649226 0.62 LMNA (0.95) MEN1KMT2AMAPTLMNACYP2D6
SCHEMBL10362320 0.62 CYP3A4 (0.42) MEN1KMT2AMAPTLMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1987009-A1 CYCLOUREA COMPOUNDS AS CALCIUM CHANNEL BLOCKERS EURO-CELTIQUE S.A. (LU) 2008-11-05 EP claimed
WO-2007085357-A1 CYCLOUREA COMPOUNDS AS CALCIUM CHANNEL BLOCKERS EURO-CELTIQUE S.A. (LU) 2007-08-02 WO claimed