SCHEMBL4656341

SCHEMBL4656341

COc1ccc(Br)c2c1CC(NC(=O)C(F)(F)F)CC2

nearest known ligand 0.57

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.57
MTNR1A P48039 10/20 0.47
MTNR1B P49286 10/20 0.47
CA1 P00915 2/20 0.45
CA2 P00918 2/20 0.45
ACHE P22303 2/20 0.45
MAPT P10636 1/20 0.45
CYP2C9 P11712 1/20 0.45
ALOX15 P16050 1/20 0.45
NQO2 P16083 1/20 0.40
ADRA1A P35348 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4216627 1.00 CYP1A2 (0.57) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4207460 0.86 MTNR1A (0.47) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4517933 0.84 MTNR1A (0.44) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4518508 0.82 MTNR1A (0.44) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4514272 0.82 MTNR1A (0.44) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4217159 0.81 MTNR1A (0.73) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL8960011 0.79 MTNR1A (0.52) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4221230 0.79 DRD4 (0.42) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL7543096 0.78 DRD2 (0.58) CYP1A2MTNR1AMTNR1BCA1CA2
SCHEMBL4519458 0.78 SMN1; SMN2 (0.51) MTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1999121-A1 NOVEL TETRALINS AS 5-HT6 MODULATORS AstraZeneca AB (SE) 2008-12-10 EP disclosed
WO-2007108742-A1 NOVEL TETRALINS AS 5-HT6 MODULATORS ASTRAZENECA AB (SE) 2007-09-27 WO disclosed