SCHEMBL4657473

SCHEMBL4657473

O=C(N1CCCC1)N(c1ccccc1)c1cc[nH]n1

nearest known ligand 0.58

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.58
POLB P06746 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
KMT2A Q03164 4/20 0.46
L3MBTL1 Q9Y468 1/20 0.44
TACR1 P25103 1/20 0.42
AGTR2 P50052 1/20 0.42
MEN1 O00255 3/20 0.40
SRD5A2 P31213 1/20 0.40
GAA P10253 1/20 0.40
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 1/20 0.37
CHRM4 P08173 1/20 0.37
CHRM5 P08912 1/20 0.37
CHRM1 P11229 1/20 0.37
CHRM3 P20309 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11195264 0.81 ALDH1A1 (0.83) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL11661567 0.80 ALDH1A1 (0.87) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL4869922 0.79 AVPR2 (0.46) ALDH1A1POLBSMN1; SMN2KMT2AMEN1
SCHEMBL4458935 0.78 NPSR1 (0.47) ALDH1A1POLBKMT2AL3MBTL1MEN1
SCHEMBL28367062 0.77 ALDH1A1 (0.62) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL398536 0.75 NPSR1 (0.44) ALDH1A1POLBKMT2AL3MBTL1MEN1
SCHEMBL6905225 0.75 KMT2A (0.46) ALDH1A1POLBKMT2AL3MBTL1MEN1
SCHEMBL3424139 0.74 SMN1; SMN2 (0.44) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL7467929 0.74 ALDH1A1 (0.77) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL402771 0.73 NPSR1 (0.41) ALDH1A1POLBKMT2AL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1917258-A2 PYRIMIDINYL-PYRAZOLE INHIBITORS OF AURORA KINASES SmithKline Beecham Corporation (US) 2008-05-07 EP disclosed
WO-2007024843-A2 PYRIMIDINYL-PYRAZOLE INHIBITORS OF AURORA KINASES SMITHKLINE BEECHAM CORPORATION (US) 2007-03-01 WO disclosed