SCHEMBL7467929

SCHEMBL7467929

O=C(N1CCN(C(=O)N(c2ccccc2)c2ccccc2)CC1)N(c1ccccc1)c1ccccc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.77
POLB P06746 1/20 0.77
SMN1; SMN2 Q16637 1/20 0.77
KMT2A Q03164 3/20 0.72
L3MBTL1 Q9Y468 1/20 0.68
AGTR2 P50052 1/20 0.65
TACR1 P25103 1/20 0.64
MEN1 O00255 2/20 0.60
GAA P10253 2/20 0.60
SRD5A2 P31213 1/20 0.56
NPSR1 Q6W5P4 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11195264 0.92 ALDH1A1 (0.83) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL10670574 0.91 ALDH1A1 (0.66) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL11661567 0.90 ALDH1A1 (0.87) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL10666586 0.89 ALDH1A1 (0.65) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL21311838 0.89 ALDH1A1 (0.69) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL7388960 0.87 ALDH1A1 (0.61) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL13182624 0.87 ALDH1A1 (0.61) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL3310703 0.87 ALDH1A1 (0.61) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL10669910 0.85 ALDH1A1 (0.59) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1
SCHEMBL14280331 0.84 ACHE (0.58) ALDH1A1POLBSMN1; SMN2KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5344830-A Anitinflammatory, cardiovascular, analgesic, central nervous system MERCK & CO., INC. (US) 1994-09-06 US disclosed
WO-1994013646-A1 N,N-DIACYLPIPERAZINE TACHYKININ ANTAGONISTS MERCK & CO., INC. (US) 1994-06-23 WO disclosed
US-5292726-A N,N-diacylpiperazines MERCK & CO., INC. (US) 1994-03-08 US disclosed
WO-1992020661-A1 N, N-DIACYLPIPERAZINES MERCK & CO., INC. (US) 1992-11-26 WO disclosed