SCHEMBL4657662

SCHEMBL4657662

CCc1cc2cc(Cl)ccc2n1S(=O)(=O)c1ccccc1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.70
PPARA Q07869 13/20 0.70
PPARD Q03181 10/20 0.70
ACLY P53396 2/20 0.47
NOD2 Q9HC29 1/20 0.46
NOD1 Q9Y239 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16486237 0.88 PPARG (0.71) PPARGPPARAPPARDACLY
SCHEMBL16486365 0.86 PPARG (0.73) PPARGPPARAPPARDACLY
SCHEMBL549089 0.84 CA12 (0.51) PPARGPPARAPPARDNOD2NOD1
SCHEMBL3562156 0.83 PPARG (0.61) PPARGPPARAPPARDACLYNOD2
SCHEMBL3520004 0.82 PPARG (1.00) PPARGPPARAPPARD
SCHEMBL3525018 0.82 PPARG (1.00) PPARGPPARAPPARD
SCHEMBL3519998 0.81 PPARG (0.98) PPARGPPARAPPARD
SCHEMBL3527488 0.80 PPARG (1.00) PPARGPPARAPPARD
SCHEMBL3520000 0.80 PPARG (0.83) PPARGPPARAPPARD
SCHEMBL3522355 0.80 PPARG (1.00) PPARGPPARAPPARDACLY

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-100482223-C As 5-HT6And/or 5-HT75-halo-tryptamine derivatives of ligands of 5-hydroxytryptamine receptors SIGMA TAU INDUSTIE FARMACEUTI (IT) 2009-04-29 CN disclosed
EP-1404317-B1 5-HALO-TRYPTAMINE DERIVATIVES USED AS LIGANDS OF THE 5-HT 6? AND/OR 5-HT 7? SEROTONIN RECEPTORS SIGMA TAU IND FARMACEUTI (IT) 2008-12-10 EP disclosed
US-7098233-B2 5-halo-tryptamine derivatives used as ligands on the 5-HT6 and/or 5-HT7 serotonin receptors SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2006-08-29 US disclosed
US-20040235899-A1 5-halo-tryptamine derivatives used as ligands of the 5-ht6 and/or 5-ht7 serotonin receptors SIGMA-TAU INDUSTRIE FARMACEUTICHE RIUNITE S.P.A. (IT) 2004-11-25 US disclosed
CN-1535146-A 5-halo-tryptamine derivatives used as ligands of 5-HT 6 and/or 5-HT7 serotonin receptors ϣ��������ҩ��ҵ��˾ 2004-10-06 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040235899-A1 5-halo-tryptamine derivatives used as ligands of the 5-ht6 and/or 5-ht7 serotonin receptors HTR7, HTR6, HTR1A PPARG 1880/4885PPARA 2380/4885PPARD 2036/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.