SCHEMBL4658445

SCHEMBL4658445

CC(C)c1ccc(CC(C#N)(C#N)CCC(F)(F)F)cc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.35
PYCR1 P32322 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
ESR1 P03372 1/20 0.31
ESR2 Q92731 1/20 0.31
ADRB1 P08588 1/20 0.31
PANK3 Q9H999 2/20 0.30
MAOB P27338 1/20 0.30
CACNA1G O43497 1/20 0.30
CACNA1H O95180 1/20 0.30
CNR2 P34972 1/20 0.30
KCNH2 Q12809 1/20 0.30
CACNA1I Q9P0X4 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4658860 0.82 SLC6A4 (0.39) IDO1NPC1RAB9AKMT2AESR1
SCHEMBL5001946 0.82 CYP2A6 (0.41) MEN1KMT2AESR1ESR2
SCHEMBL4657169 0.82 ESR1 (0.33) IDO1ESR1ESR2
SCHEMBL4657291 0.81
SCHEMBL4658834 0.80 MAOA (0.33) IDO1RAB9AKMT2AESR1ESR2
SCHEMBL4658745 0.79 ESR1 (0.41) ESR1ESR2KCNH2
SCHEMBL4657451 0.79 TAAR1 (0.39) IDO1PYCR1KMT2AESR1ESR2
SCHEMBL4657566 0.79 LOXL2 (0.41) IDO1NPC1RAB9AMAOBKCNH2
SCHEMBL4723541 0.79 MAOB (0.33) PYCR1ESR1ESR2MAOB
SCHEMBL4657371 0.79 ESR1 (0.32) ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 IDO1 382/4885PYCR1 402/4885NPC1 400/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 IDO1 278/4885PYCR1 272/4885NPC1 252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.