SCHEMBL4658745

SCHEMBL4658745

CC(C)(C)c1ccc(CC(C#N)(C#N)CCC(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 4/20 0.41
ESR2 Q92731 4/20 0.41
GRM2 Q14416 1/20 0.36
KIF11 P52732 1/20 0.36
EPHX2 P34913 2/20 0.35
TSHR P16473 2/20 0.33
KCNH2 Q12809 1/20 0.33
TP53 P04637 1/20 0.33
GRIA2 P42262 1/20 0.32
GRIA4 P48058 1/20 0.32
DHODH Q02127 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4657451 0.87 TAAR1 (0.39) ESR1ESR2KIF11
SCHEMBL5001946 0.83 CYP2A6 (0.41) ESR1ESR2TP53
SCHEMBL4657169 0.83 ESR1 (0.33) ESR1ESR2
SCHEMBL4658834 0.81 MAOA (0.33) ESR1ESR2
SCHEMBL4657566 0.80 LOXL2 (0.41) KIF11KCNH2
SCHEMBL4657371 0.80 ESR1 (0.32) ESR1ESR2
SCHEMBL4658860 0.80 SLC6A4 (0.39) ESR1ESR2EPHX2KCNH2
SCHEMBL4723541 0.80 MAOB (0.33) ESR1ESR2
SCHEMBL4657447 0.80 ATM (0.40) EPHX2
SCHEMBL4657428 0.79 ALDH1A1 (0.39) TSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1385817-B1 MALONONITRILE COMPOUNDS AND THEIR USE AS PESTICIDES SUMITOMO CHEMICAL CO (JP) 2008-12-03 EP disclosed
US-7402691-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2008-07-22 US disclosed
US-7011838-B2 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2006-03-14 US disclosed
US-20050209323-A1 Malononitrile compounds and their use as pesticides OTAKA KEN 2005-09-22 US disclosed
US-20040138065-A1 Malononitrile compounds and their use as pesticides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 2004-07-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209323-A1 Malononitrile compounds and their use as pesticides C1S, C1R, C5 ESR1 4561/4885ESR2 4792/4885GRM2 3240/4885
US-20040138065-A1 Malononitrile compounds and their use as pesticides CBR1, MAL2, CBR3 ESR1 4835/4885ESR2 4741/4885GRM2 2136/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.