SCHEMBL465890

SCHEMBL465890

Nc1ccc([N+](=O)[O-])cc1C(=O)CCC(N)C(=O)O

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.50
ALDH1A1 P00352 1/20 0.49
CYP3A4 P08684 1/20 0.49
ALOX15 P16050 1/20 0.49
TDP1 Q9NUW8 1/20 0.49
GRM8 O00222 10/20 0.47
GRM4 Q14833 10/20 0.47
GRM6 O15303 5/20 0.46
PTPRA P18433 1/20 0.45
CYP2C19 P33261 1/20 0.44
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9543018 1.00 KMO (0.50) KMOALDH1A1CYP3A4ALOX15TDP1
SCHEMBL639675 1.00 KMO (0.50) KMOALDH1A1CYP3A4ALOX15TDP1
Water SCHEMBL6282445 0.99 KMO (0.49) KMOALDH1A1CYP3A4ALOX15TDP1
Hydrochloric Acid SCHEMBL11310889 0.99 KMO (0.49) KMOALDH1A1CYP3A4ALOX15TDP1
Hydrochloric Acid SCHEMBL10950905 0.99 KMO (0.49) KMOALDH1A1CYP3A4ALOX15TDP1
Bromide SCHEMBL10946974 0.99 KMO (0.49) KMOALDH1A1CYP3A4ALOX15TDP1
Iodide SCHEMBL10947423 0.99 KMO (0.49) KMOALDH1A1CYP3A4ALOX15TDP1
SCHEMBL10613892 0.81 KMT2A (0.50) ALDH1A1CYP3A4ALOX15TDP1GRM8
4-Nitroaniline SCHEMBL10698315 0.81 CCR2 (0.38) KMOGRM8GRM4GRM6GAA
SCHEMBL4414897 0.80 KMT2A (0.44) ALDH1A1CYP3A4ALOX15TDP1GRM8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230220387-A1 D-SERINE TRANSPORT MODIFIER AND SCREENING METHOD THEREOF, AND SCREENING METHOD OF D-SERINE TRANSPORTER PROTEIN KAGAMI INC. (JP) 2023-07-13 US claimed
US-9611502-B2 Method for simultaneously measuring activity of various enzymes by using multi-wavelength absorption single channel CHONGQING MEDICAL UNIVERSITY (CN) 2017-04-04 US claimed
US-20150225764-A1 METHOD FOR SIMULTANEOUSLY MEASURING ACTIVITY OF VARIOUS ENZYMES BY USING MULTI-WAVELENGTH ABSORPTION SINGLE CHANNEL CHONGQING MEDICAL UNIVERSITY (CN) 2015-08-13 US claimed
US-8486650-B2 Method of detecting serum gamma-glutamyl transferase isoforms in a biological fluid UNIVERSITA' DI PISA (IT) 2013-07-16 US claimed
US-20110016582-A1 Biosynthetic Engineering of Glucosinolates UNIVERSITY OF COPENHAGEN (DK) 2011-01-20 US claimed
EP-2257630-A2 BIOSYNTHETIC ENGINEERING OF GLUCOSINOLATES University of Copenhagen (DK) 2010-12-08 EP claimed
US-20100227351-A1 METHOD OF DETECTING AND SEPARATING SERUM GAMMA-GLUTAMYL TRANSFERASE (GGT) ISOFORMS IN A SAMPLE OF BIOLOGICAL FLUID AND THE ENZYME ISOFORMS THEREBY OBTAINED UNIVERSITA' DI PISA (IT) 2010-09-09 US claimed
WO-2009106985-A2 BIOSYNTHETIC ENGINEERING OF GLUCOSINOLATES UNIVERSITY OF COPENHAGEN (DK) 2009-09-03 WO claimed
EP-0207406-B1 REAGENT SHEET AND INTEGRAL MULTILAYER ANALYTICAL ELEMENT FOR MEASUREMENT OF GAMMA-GLUTAMYL TRANSFERASE ACTIVITY FUJI PHOTO FILM CO., LTD. (JP) 1993-03-10 EP claimed
US-4916059-A GAMMA-GLUTAMYL TRANSFERASE FUJI PHOTO FILM CO., LTD. (JP) 1990-04-10 US claimed
US-4511651-A Reagent composition and assay for the determination of γ-glutamyltransferase activity AMERICAN MONITOR CORPORATION (US) 1985-04-16 US claimed
US-4372874-A Stabilization of hydrolysis prone labile organic reagents in liquid media MEDICAL ANALYSIS SYSTEMS, INC. 1983-02-08 US claimed
US-4049702-A DIAGNOSIS OF LIVER DISEASE BY DETERMINATION OF G-GLUTAMYL-TRANS-PEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1977-09-20 US claimed
US-3986931-A γ-GLUTAMYL-4-NITROANILIDE COMPOUNDS AND THEIR USE IN DETERMINING γ-GLUTAMYL TRANSPEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1976-10-19 US claimed
US-3979447-A DETERMINATION OF G-GLUTAMYLTRANSPEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1976-09-07 US claimed
JP-10108694-A None JP disclosed
JP-9071514-A None JP disclosed
US-3979447-A DETERMINATION OF G-GLUTAMYLTRANSPEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1976-09-07 US disclosed
US-3979447-A DETERMINATION OF G-GLUTAMYLTRANSPEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1976-09-07 US disclosed
US-3979447-A DETERMINATION OF G-GLUTAMYLTRANSPEPTIDASE BOEHRINGER MANNHEIM G.M.B.H. (DT) 1976-09-07 US disclosed