SCHEMBL4659111

SCHEMBL4659111

O=S(=O)(Nc1c[nH]cn1)c1cncs1

nearest known ligand 0.34

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.34
KDM4E B2RXH2 3/20 0.33
KAT7 O95251 1/20 0.32
KAT6A Q92794 1/20 0.32
KAT5 Q92993 1/20 0.32
KAT8 Q9H7Z6 1/20 0.32
KMT2A Q03164 2/20 0.31
MAPT P10636 1/20 0.31
GAA P10253 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27624078 0.65 HPGD (0.36) ALDH1A1KDM4EKMT2AMAPTGAA
SCHEMBL4659266 0.64 ABCC9 (0.40) ALDH1A1KDM4EKAT7KAT6AKAT5
SCHEMBL3854458 0.63 ALDH1A1 (0.50) ALDH1A1KDM4EKMT2AGAA
SCHEMBL23124196 0.63 IMPDH2 (0.37)
SCHEMBL8560391 0.62 TDP1 (0.40) ALDH1A1KDM4EKAT7KAT6AKAT5
SCHEMBL27785439 0.62 KAT7 (0.37) KAT7KAT6AKAT5KAT8KMT2A
SCHEMBL9095381 0.60 NAMPT (0.34)
SCHEMBL10044450 0.60 RXFP1 (0.59) ALDH1A1KDM4EKMT2AMAPTGAA
SCHEMBL3857993 0.60 ALDH1A1 (0.64) ALDH1A1KMT2AMAPT
Hydrochloric Acid SCHEMBL27576989 0.59 HDAC8 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2001849-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. Hoffmann-Roche AG (CH) 2008-12-17 EP disclosed
WO-2007110337-A1 PYRIDINE AND PYRIMIDINE DERIVATIVES AS MGLUR2 ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2007-10-04 WO disclosed