SCHEMBL4662765

SCHEMBL4662765

Cc1ccccc1Nc1ccc(CN(C)c2ccccc2C(C)O)cc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.38
CDK2 P24941 2/20 0.38
MAPK13 O15264 1/20 0.35
MAPK12 P53778 1/20 0.35
MAPK11 Q15759 1/20 0.35
MAPK14 Q16539 1/20 0.35
HTT P42858 1/20 0.34
LIMK2 P53671 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
ITGB1 P05556 3/20 0.32
ITGA4 P13612 3/20 0.32
NR3C1 P04150 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661488 0.89 HTT (0.40) HTTALDH1A1
SCHEMBL4661449 0.87 CDK4 (0.38) CDK4CDK2HTTKDM4EALDH1A1
SCHEMBL4661583 0.87 CDK4 (0.38) CDK4CDK2HTTKDM4EALDH1A1
SCHEMBL4661500 0.86 ALDH1A1 (0.41) HTTLIMK2KDM4EALDH1A1
SCHEMBL4661323 0.86 ALDH1A1 (0.41) HTTLIMK2KDM4EALDH1A1
SCHEMBL4661434 0.82 CDK4 (0.40) CDK4CDK2KDM4E
SCHEMBL4661305 0.76 PYCR1 (0.42) HTTKDM4EALDH1A1
SCHEMBL4661399 0.76 PYCR1 (0.42) HTTKDM4EALDH1A1
SCHEMBL4346610 0.74 KDM4E (0.55) CDK4CDK2MAPK13MAPK12MAPK11
SCHEMBL4661242 0.73 POLB (0.45) CDK4CDK2HTTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007707-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2008-12-31 EP disclosed
WO-2007118041-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-10-18 WO disclosed