SCHEMBL4661583

SCHEMBL4661583

CC(O)c1ccccc1N(C)Cc1ccc(Nc2ccccc2Cl)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK4 P11802 2/20 0.38
CDK2 P24941 2/20 0.38
CCNE1 P24864 1/20 0.38
ADRB2 P07550 2/20 0.37
ADRB1 P08588 2/20 0.37
AOC3 Q16853 1/20 0.37
CYP2D6 P10635 2/20 0.36
NFKB1 P19838 1/20 0.36
HIF1A Q16665 1/20 0.36
ALDH1A1 P00352 3/20 0.36
BLM P54132 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4661449 1.00 CDK4 (0.38) CDK4CDK2CCNE1ADRB2ADRB1
SCHEMBL4661434 0.88 CDK4 (0.40) CDK4CDK2BLMCYP1A2CYP2C19
SCHEMBL4662765 0.87 CDK4 (0.38) CDK4CDK2ALDH1A1HTTKDM4E
SCHEMBL4661323 0.85 ALDH1A1 (0.41) HIF1AALDH1A1SMN1; SMN2CYP3A4MEN1
SCHEMBL4661500 0.85 ALDH1A1 (0.41) HIF1AALDH1A1SMN1; SMN2CYP3A4MEN1
SCHEMBL4662702 0.83 JAK2 (0.42) CDK4CDK2CCNE1ADRB2ADRB1
SCHEMBL4661488 0.81 HTT (0.40) ALDH1A1SMN1; SMN2MEN1KMT2AHTT
SCHEMBL4661452 0.79 CXCL8 (0.36) CDK4CDK2CCNE1CYP2D6ALDH1A1
SCHEMBL4661305 0.75 PYCR1 (0.42) ALDH1A1SMN1; SMN2MEN1KMT2AL3MBTL1
SCHEMBL4661399 0.75 PYCR1 (0.42) ALDH1A1SMN1; SMN2MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007707-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR Boehringer Ingelheim International GmbH (DE) 2008-12-31 EP disclosed
WO-2007118041-A1 COMPOUNDS WHICH MODULATE THE CB2 RECEPTOR BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-10-18 WO disclosed