SCHEMBL4664513

SCHEMBL4664513

CCCOCc1ccc(C#N)cn1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
HPGD P15428 2/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
HTT P42858 1/20 0.46
MBOAT4 Q96T53 1/20 0.41
CYP2A6 P11509 1/20 0.35
GABRA5 P31644 1/20 0.34
HPGDS O60760 1/20 0.34
MAOB P27338 1/20 0.33
MAPT P10636 1/20 0.33
FNTA P49354 1/20 0.33
FNTB P49356 1/20 0.33
PGGT1B P53609 1/20 0.33
RORC P51449 1/20 0.33
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30832037 0.87 MBOAT4 (0.43) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL1145890 0.80 KDM4E (0.42) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL7219997 0.78 CYP19A1 (0.45) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL2633134 0.77 CYP2A6 (0.48) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL10263917 0.76 SYK (0.40) ALDH1A1KDM4EHPGDL3MBTL1GABRA5
SCHEMBL13141087 0.76 MBOAT4 (0.42) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL1145885 0.76 MBOAT4 (0.39) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL2578930 0.75 MBOAT4 (0.40) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL19387952 0.75 RORC (0.40) ALDH1A1KDM4EHPGDL3MBTL1HTT
SCHEMBL7433167 0.75 ALDH1A1 (0.49) ALDH1A1KDM4EHPGDL3MBTL1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1924561-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS Eli Lilly & Company (US) 2008-05-28 EP disclosed
WO-2007028083-A2 6-ARYLALKYLAMINO- 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2007-03-08 WO disclosed