SCHEMBL4664691

SCHEMBL4664691

CCc1cc(Nc2ccc(C)cc2C(=O)O)n(-c2ncccc2C)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 1/20 0.43
LMNA P02545 2/20 0.42
GAA P10253 1/20 0.42
DHODH Q02127 13/20 0.42
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 1/20 0.39
MAPT P10636 1/20 0.39
RAB9A P51151 1/20 0.39
KDM5A P29375 1/20 0.39
KDM4C Q9H3R0 1/20 0.39
KDM5B Q9UGL1 1/20 0.39
MYC P01106 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600206 0.88 ADORA1 (0.42) ADORA1DHODHKDM5AKDM4CKDM5B
SCHEMBL14600232 0.85 DHODH (0.46) ADORA1LMNADHODHMEN1KMT2A
SCHEMBL14600465 0.84 DHODH (0.46) ADORA1DHODHMAPT
SCHEMBL14600450 0.81 DHODH (0.43) ADORA1DHODHMAPT
SCHEMBL14600229 0.80 ADORA1 (0.45) ADORA1LMNAGAADHODH
SCHEMBL14600441 0.78 ADORA1 (0.56) ADORA1DHODH
SCHEMBL14600727 0.78 DHODH (0.55) ADORA1DHODHMEN1KMT2AHTT
SCHEMBL14600498 0.78 DHODH (0.42) ADORA1DHODHMAPT
SCHEMBL14600231 0.78 SORT1 (0.50) LMNAGAAMEN1KMT2ANPC1
SCHEMBL14600468 0.78 DHODH (0.40) ADORA1LMNAGAADHODHMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed