SCHEMBL4665241

SCHEMBL4665241

Cc1ccc(Nc2cc(-c3cccc(OC(C)C)c3)nn2-c2sccc2C)c(C(=O)O)c1

nearest known ligand 0.54

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 13/20 0.54
KEAP1 Q14145 1/20 0.39
NFE2L2 Q16236 1/20 0.39
MAPT P10636 2/20 0.38
TP53 P04637 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14600273 0.93 DHODH (0.46) DHODHKEAP1NFE2L2MAPTTP53
SCHEMBL4666640 0.85 DHODH (0.58) DHODHKEAP1NFE2L2MAPTTP53
Hydrochloric Acid SCHEMBL4666221 0.84 DHODH (0.57) DHODHKEAP1NFE2L2MAPTTP53
SCHEMBL14600682 0.80 DHODH (0.55) DHODHKEAP1NFE2L2
SCHEMBL4668988 0.77 DHODH (0.49) DHODHKEAP1NFE2L2MAPTTP53
SCHEMBL5008553 0.77 ADORA1 (0.59) DHODHMAPTTP53
SCHEMBL14600673 0.76 DHODH (0.47) DHODHKEAP1NFE2L2MAPTTP53
SCHEMBL14600691 0.75 DHODH (0.49) DHODHKEAP1NFE2L2
SCHEMBL4666815 0.75 ALDH1A1 (0.42) KEAP1NFE2L2MAPTTP53FABP3
SCHEMBL14600727 0.75 DHODH (0.55) DHODH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed