SCHEMBL4665768

SCHEMBL4665768

Cc1ccc(S(=O)(=O)Nc2ccc(Nc3cc(-c4cccc(C(F)(F)F)c4C(F)(F)F)ncn3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNNI3K Q59H18 2/20 0.46
FFAR4 Q5NUL3 2/20 0.46
CDK1 P06493 2/20 0.45
CCNB1 P14635 2/20 0.45
CDK7 P50613 2/20 0.45
CCNH P51946 2/20 0.45
FFAR1 O14842 1/20 0.45
CCNA2 P20248 1/20 0.45
CDK2 P24941 1/20 0.45
CCNA1 P78396 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.44
CCNT1 O60563 3/20 0.44
CDK9 P50750 3/20 0.44
CYP1A2 P05177 3/20 0.43
CYP3A4 P08684 3/20 0.43
CYP2D6 P10635 2/20 0.43
MAPK1 P28482 2/20 0.43
CYP2C19 P33261 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4667473 0.81 MEN1 (0.51) TNNI3KCDK1CCNB1CDK7CCNH
SCHEMBL4663808 0.79 ALDH1A1 (0.54) TNNI3KMEN1KMT2AGAACCNT1
SCHEMBL4098710 0.79 CDK9 (0.64) CDK1CCNB1CDK7CCNHCCNA2
SCHEMBL4665854 0.78 BACE1 (0.60) TNNI3KFFAR1MEN1KMT2AGAA
SCHEMBL17352240 0.76 CCNT1 (0.66) MEN1KMT2ACCNT1CDK9CYP1A2
SCHEMBL4666121 0.76 MEN1 (0.45) TNNI3KCDK1CCNB1CDK7CCNH
SCHEMBL4664257 0.75 CCNT1 (0.64) TNNI3KMEN1KMT2AGAACCNT1
SCHEMBL3397888 0.75 ABL1 (0.74) MAPK1TP53MAPTABL1BCR
SCHEMBL4666152 0.75 ABL1 (0.74) MAPK1TP53MAPTABL1BCR
SCHEMBL4665837 0.75 SLC22A12 (0.50) CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors ALTANA PHARMA AG (DE) 2008-10-02 US claimed
EP-1709007-A1 N-4-(6-(HETEO)ARYL-PYRIMIDIN-4-YLAMINOPHENYL)-BENZENESULFONAMIDES AS KINASE INHIBITORS Altana Pharma AG (DE) 2006-10-11 EP claimed
WO-2005070900-A1 N-4-(6- (HETEO) ARYL-PYRIMIDIN-4-YLAMINOPHENYL) -BEZENESULFONAMIDES AS KINASE INHIBITORS ALTANA PHARMA AG (DE) 2005-08-04 WO claimed
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors ALTANA PHARMA AG (DE) 2008-10-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242681-A1 N-4-(6-(Hetero)Aryl-Pyrimidin-4-Ylaminophenyl)-Benzenesulfonamides as Kinase Inhibitors MAP3K19, MAP3K6, MAP3K20 TNNI3K 25/4885FFAR4 1779/4885CDK1 68/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.