SCHEMBL4666107

SCHEMBL4666107

CS(=O)(=O)Nc1ccc(-c2ccc(O)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 5/20 0.66
UQCRB P14927 1/20 0.56
DYRK1B Q9Y463 2/20 0.56
CLK1 P49759 1/20 0.56
DYRK1A Q13627 1/20 0.56
DYRK2 Q92630 1/20 0.56
HSD17B1 P14061 1/20 0.55
HSD17B2 P37059 1/20 0.55
CA1 P00915 2/20 0.55
CA2 P00918 2/20 0.55
KEAP1 Q14145 1/20 0.54
HPGD P15428 3/20 0.53
ALDH1A1 P00352 3/20 0.53
SMN1; SMN2 Q16637 2/20 0.53
KDM4E B2RXH2 1/20 0.53
LMNA P02545 1/20 0.53
HTT P42858 1/20 0.53
CA12 O43570 1/20 0.52
CA9 Q16790 1/20 0.52
USP7 Q93009 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL518114 0.94 CA1 (0.61) KIF11UQCRBCA1CA2KEAP1
SCHEMBL19227700 0.89 LMNA (0.57) KIF11UQCRBDYRK1BCLK1DYRK1A
SCHEMBL31041151 0.89 KIF11 (0.79) KIF11DYRK1AHSD17B1HSD17B2CA1
Lithium SCHEMBL31041154 0.87 KIF11 (0.76) KIF11DYRK1AHSD17B1HSD17B2CA1
SCHEMBL12054668 0.82 KEAP1 (0.75) KIF11CA1CA2KEAP1HPGD
SCHEMBL21254711 0.81 KIF11 (0.68) KIF11DYRK1AHSD17B1HSD17B2CA1
SCHEMBL873846 0.81 KEAP1 (0.75) KIF11UQCRBCA1CA2KEAP1
SCHEMBL4661398 0.81 KIF11 (0.68) KIF11DYRK1AHSD17B1HSD17B2CA1
SCHEMBL15771505 0.80 KIF11 (0.62) KIF11HSD17B1HSD17B2CA1CA2
SCHEMBL2497654 0.79 KIF11 (0.66) KIF11DYRK1AHSD17B1HSD17B2CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1193250-B1 PHENYL SULFAMATE DERIVATIVES TEIKOKU HORMONE MFG CO LTD (JP) 2008-06-04 EP disclosed
US-6762205-B1 STEROID SULFATASE INHIBITORS WITHOUT ESTROGENIC SIDE EFFECT ACTION TEIKOKU HORMONE MFG. CO., LTD. (JP) 2004-07-13 US disclosed
EP-1193250-A1 PHENYL SULFAMATE DERIVATIVES Teikoku Hormone Mfg. Co., Ltd. (JP) 2002-04-03 EP disclosed