SCHEMBL4666247

SCHEMBL4666247

CCc1nn(-c2nc(C)cnc2C)c(Nc2ccc(C)cc2C(=O)OC)c1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
RXFP1 Q9HBX9 1/20 0.36
HCRTR1 O43613 2/20 0.34
HCRTR2 O43614 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
TP53 P04637 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
DHODH Q02127 2/20 0.33
ALDH1A1 P00352 1/20 0.32
HPGD P15428 1/20 0.32
AHR P35869 1/20 0.32
OPRK1 P41145 2/20 0.32
TSHR P16473 2/20 0.32
MAPT P10636 1/20 0.32
ADORA1 P30542 3/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4666119 0.83 ADORA1 (0.39) HCRTR1HCRTR2SMN1; SMN2MEN1KMT2A
SCHEMBL14600228 0.81 HPGD (0.38) NPC1RAB9ARXFP1HCRTR1HCRTR2
SCHEMBL14600247 0.77 ADORA1 (0.43) DHODHADORA1
SCHEMBL14600448 0.75 ADORA1 (0.43) DHODHALDH1A1HPGDADORA1
SCHEMBL14600435 0.75 ADORA1 (0.45) DHODHADORA1
SCHEMBL14600229 0.73 ADORA1 (0.45) DHODHADORA1
SCHEMBL4665671 0.72 P2RY1 (0.37) TP53DHODHMAPTADORA1
SCHEMBL14600450 0.71 DHODH (0.43) HCRTR1HCRTR2DHODHMAPTADORA1
SCHEMBL4666602 0.71 ADORA1 (0.39) RXFP1MAPTADORA1
SCHEMBL4668860 0.70 KCNMA1 (0.38) NPC1RXFP1TP53MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1928455-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES Bayer Healthcare, LLC (US) 2008-06-11 EP disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed
WO-2007027842-A1 ANILINOPYRAZOLE DERIVATIVES USEFUL FOR THE TREATMENT OF DIABETES BAYER HEALTHCARE LLC (US) 2007-03-08 WO disclosed