SCHEMBL4666734

SCHEMBL4666734

CC(C)COC(=O)N1CCC(c2c[nH]c3c(C(N)=O)nc(-c4ccccc4)cc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 16/20 0.48
CHUK O15111 5/20 0.48
AURKA O14965 1/20 0.46
FLT3 P36888 1/20 0.46
CSNK1E P49674 1/20 0.46
BTK Q06187 1/20 0.46
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
GPR119 Q8TDV5 1/20 0.40
JAK2 O60674 1/20 0.40
TLR9 Q9NR96 1/20 0.39
TLR8 Q9NR97 1/20 0.39
TLR7 Q9NYK1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5011762 0.85 IKBKB (0.48) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL4664992 0.85 ALDH1A1 (0.41) KDM4EALDH1A1HPGDHSD17B10GPR119
SCHEMBL5786506 0.83 IKBKB (0.66) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL4666771 0.82 JAK2 (0.52) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL4664932 0.82 IKBKB (0.70) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL14048291 0.80 IKBKB (0.54) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL4665003 0.80 JAK2 (0.38) AURKAFLT3BTKJAK2
SCHEMBL4664929 0.78 IKBKB (0.65) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL5785013 0.76 IKBKB (0.56) IKBKBCHUKAURKAFLT3CSNK1E
SCHEMBL5024842 0.76 IKBKB (0.47) IKBKBCHUKAURKAFLT3CSNK1E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940296-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-07-09 EP claimed
WO-2007114848-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-11 WO claimed
EP-1940296-A2 CHEMICAL COMPOUNDS SmithKline Beecham Corporation (US) 2008-07-09 EP disclosed
WO-2007114848-A2 CHEMICAL COMPOUNDS SMITHKLINE BEECHAM CORPORATION (US) 2007-10-11 WO disclosed