SCHEMBL4667074

SCHEMBL4667074

CCN(C(=O)c1c(CN2CCN(C)CC2)c(-c2ccccc2)nc2ccccc12)c1ccccc1C#N

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 14/20 0.53
KCNH2 Q12809 6/20 0.53
TACR2 P21452 8/20 0.47
OPRM1 P35372 4/20 0.45
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
TSHR P16473 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668624 0.85 TACR3 (0.38) TACR3KCNH2TACR2KDM4EALDH1A1
SCHEMBL4668567 0.79 TACR3 (0.37) TACR3TACR2OPRM1KDM4EALDH1A1
SCHEMBL4667075 0.78 TACR3 (0.57) TACR3KCNH2TACR2OPRM1
SCHEMBL4668577 0.77 TACR3 (0.36) TACR3KCNH2TACR2OPRM1KDM4E
SCHEMBL28773315 0.76 TACR3 (0.55) TACR3KCNH2TACR2OPRM1
SCHEMBL4667051 0.75 TACR3 (0.55) TACR3KCNH2TACR2OPRM1
SCHEMBL6996763 0.74 TACR3 (0.54) TACR3KCNH2TACR2OPRM1
SCHEMBL6266946 0.72 TACR2 (0.59) TACR3KCNH2TACR2OPRM1TSHR
SCHEMBL6848956 0.72 TACR2 (0.61) TACR3KCNH2TACR2OPRM1TSHR
SCHEMBL6853049 0.71 TACR3 (0.58) TACR3KCNH2TACR2OPRM1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940795-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-07-09 EP disclosed
WO-2007035156-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO disclosed