SCHEMBL4668568

SCHEMBL4668568

N#Cc1ccccc1CCNC(=O)c1c(C[N+]2([O-])CCCC2)c(-c2ccccc2)nc2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.50
TP53 P04637 2/20 0.41
TACR3 P29371 9/20 0.40
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
TACR2 P21452 4/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HIF1A Q16665 1/20 0.37
OPRM1 P35372 1/20 0.37
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668578 0.92 LMNA (0.48) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4668628 0.91 LMNA (0.49) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4665273 0.86 LMNA (0.67) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4665278 0.85 LMNA (0.66) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4665602 0.83 LMNA (0.57) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4668637 0.83 LMNA (0.59) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4665270 0.82 LMNA (0.58) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4667328 0.81 LMNA (0.53) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL4668727 0.81 LMNA (0.53) LMNATP53TACR3ALDH1A1HPGD
SCHEMBL5042219 0.81 LMNA (0.55) LMNATP53TACR3ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940795-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-07-09 EP disclosed
WO-2007035156-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO disclosed