SCHEMBL4668628

SCHEMBL4668628

CN1CC[N+]([O-])(Cc2c(-c3ccccc3)nc3ccccc3c2C(=O)NCCc2ccccc2C#N)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
TACR3 P29371 8/20 0.41
KCNH2 Q12809 1/20 0.41
TP53 P04637 1/20 0.40
TACR2 P21452 5/20 0.39
OPRM1 P35372 1/20 0.38
ALDH1A1 P00352 1/20 0.37
HPGD P15428 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4668568 0.91 LMNA (0.50) LMNATACR3KCNH2TP53TACR2
SCHEMBL4668578 0.89 LMNA (0.48) LMNATACR3KCNH2TP53TACR2
SCHEMBL4665275 0.87 LMNA (0.64) LMNATACR3KCNH2TP53TACR2
SCHEMBL4667075 0.85 TACR3 (0.57) LMNATACR3KCNH2TACR2OPRM1
SCHEMBL4665243 0.84 LMNA (0.57) LMNATACR3KCNH2TP53TACR2
SCHEMBL4667069 0.80 TACR3 (0.47) LMNATACR3KCNH2TACR2OPRM1
SCHEMBL4665602 0.80 LMNA (0.57) LMNATACR3TP53TACR2OPRM1
SCHEMBL5042219 0.80 LMNA (0.55) LMNATACR3TP53TACR2OPRM1
SCHEMBL5045996 0.79 LMNA (0.57) LMNATACR3TP53TACR2OPRM1
SCHEMBL4668624 0.79 TACR3 (0.38) TACR3KCNH2TACR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1940795-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS AstraZeneca AB (SE) 2008-07-09 EP claimed
WO-2007035156-A1 N-OXO-HETEROCYCLE AND N-OXO-ALKYL QUINOLINE-4-CARBOXAMIDES AS NK-3 RECEPTOR LIGANDS ASTRAZENECA AB (SE) 2007-03-29 WO claimed