SCHEMBL4670514

SCHEMBL4670514

C=CCn1c(=O)c2c(nc(C#Cc3cccc(C)c3)n2C)n(C)c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.56
ALDH1A1 P00352 2/20 0.56
HTT P42858 2/20 0.52
HSD17B10 Q99714 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MAPT P10636 1/20 0.48
THRB P10828 1/20 0.48
HPGD P15428 1/20 0.48
BLM P54132 1/20 0.48
RCE1 Q9Y256 1/20 0.48
TP53 P04637 1/20 0.47
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
PKM P14618 2/20 0.43
TTR P02766 1/20 0.42
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4637292 0.89 ADORA2B (0.53) ADORA2BALDH1A1HSD17B10KDM4EMAPT
SCHEMBL4636001 0.87 MAOA (0.43) ALDH1A1HTTMAPTTHRBLMNA
SCHEMBL4636778 0.87 ADORA2B (0.51) ADORA2BALDH1A1HTTHSD17B10KDM4E
SCHEMBL2542730 0.84 ADORA2B (0.46) ADORA2BBLM
SCHEMBL4668176 0.81 PDE5A (0.40) ALDH1A1HTTMAPTTHRBLMNA
SCHEMBL4636158 0.81 ADORA1 (0.48) ADORA2BCYP2C9
SCHEMBL2542959 0.76 ADORA2A (0.43) ADORA2B
SCHEMBL4636790 0.76 MAOB (0.47) ADORA2BALDH1A1HSD17B10KDM4EHPGD
SCHEMBL2537917 0.76 ADORA1 (0.45) ADORA2BBLM
SCHEMBL2540207 0.75 ADORA1 (0.53) ADORA2BHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed