SCHEMBL4668176

SCHEMBL4668176

Cc1cccc(C#Cc2nc3c(c(=O)n(CC4CCC4)c(=O)n3C)n2C)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 2/20 0.40
PDE4A P27815 2/20 0.40
PDE4B Q07343 2/20 0.40
PDE4C Q08493 2/20 0.40
PDE4D Q08499 2/20 0.40
MAPT P10636 3/20 0.40
NPSR1 Q6W5P4 2/20 0.40
ALDH1A1 P00352 2/20 0.40
ALOX12 P18054 1/20 0.40
HTT P42858 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
THRB P10828 3/20 0.39
POLB P06746 2/20 0.39
MAOA P21397 4/20 0.39
MAOB P27338 4/20 0.39
MAPK1 P28482 1/20 0.39
LMNA P02545 1/20 0.38
TSHR P16473 1/20 0.38
ADORA2A P29274 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4636762 0.90 MAOB (0.41) PDE5APDE4APDE4BPDE4CPDE4D
SCHEMBL4636001 0.85 MAOA (0.43) MAPTNPSR1ALDH1A1ALOX12HTT
SCHEMBL2542730 0.82 ADORA2B (0.46) MAOBADORA2AADORA1
SCHEMBL4670514 0.81 ADORA2B (0.56) MAPTALDH1A1HTTTHRBPOLB
SCHEMBL4636158 0.79 ADORA1 (0.48) PDE4APDE4DADORA3MAOBADORA2A
SCHEMBL4636591 0.76 ADORA1 (0.54) ADORA3MAOBADORA2AADORA1
SCHEMBL2542959 0.74 ADORA2A (0.43) ADORA2AADORA1
SCHEMBL4636790 0.74 MAOB (0.47) ALDH1A1POLBMAOAMAOBADORA2A
SCHEMBL4636217 0.73 ADORA3 (0.47) ALDH1A1HTTADORA3POLBMAOA
SCHEMBL4637264 0.72 MAOB (0.47) MAPTALDH1A1ADORA3MAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1939197-A1 8-ethinylxanthine derivatives as selective A2A receptor antagonists SCHWARZ PHARMA AG (DE) 2008-07-02 EP disclosed