SCHEMBL4673725

SCHEMBL4673725

CCCCc1oc2ccccc2c1OC(=O)N(C)CCc1ccc2cc(OCc3nnn[nH]3)ccc2c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 1/20 0.41
PTPN1 P18031 7/20 0.41
SIRT3 Q9NTG7 4/20 0.38
PPARG P37231 4/20 0.37
PPARA Q07869 4/20 0.37
PPARD Q03181 2/20 0.37
ALDH1A1 P00352 2/20 0.36
TP53 P04637 2/20 0.36
CYP3A4 P08684 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
THRA P10827 2/20 0.36
THRB P10828 2/20 0.36
KDM5A P29375 2/20 0.36
KDM7A Q6ZMT4 2/20 0.36
MLNR O43193 1/20 0.36
CACNA1F O60840 1/20 0.36
PHF2 O75151 1/20 0.36
ABCB11 O95342 1/20 0.36
NR3C1 P04150 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4674314 0.89 NR1H4 (0.48) NR1H4PTPN1SIRT3PPARGPPARA
SCHEMBL4728486 0.86 NR1H4 (0.42) NR1H4PTPN1SIRT3THRATHRB
SCHEMBL4672473 0.82 PTPN1 (0.51) NR1H4PTPN1SIRT3
SCHEMBL4674317 0.80 NR1H4 (0.49) NR1H4PTPN1SIRT3ALDH1A1TP53
SCHEMBL4672520 0.78 PTPN1 (0.50) NR1H4PTPN1SIRT3ALDH1A1TP53
SCHEMBL4674079 0.77 PTPN1 (0.52) NR1H4PTPN1SIRT3SMN1; SMN2THRA
SCHEMBL4673738 0.75 PTPN1 (0.52) NR1H4PTPN1SIRT3ABCB1
SCHEMBL4674024 0.74 PTPN1 (0.43) NR1H4PTPN1SMN1; SMN2MEN1MAPT
SCHEMBL4670614 0.74 PTPN1 (0.39) NR1H4PTPN1SIRT3KDM7AMAPT
SCHEMBL4670309 0.74 PTPN1 (0.43) NR1H4PTPN1SIRT3THRATHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1397341-B1 6-(ARYL-AMIDO OR ARYL-AMIDOMETHYL)-NAPHTHALEN-2-YLOXY-ACIDIC DERIVATIVES AS INHIBITORS OF PLASMINOGEN ACTIVATOR INHIBITOR TYPE-1 (PAI-1) WYETH CORP (US) 2008-08-06 EP claimed