SCHEMBL4674060

SCHEMBL4674060

O=C(O)c1c(F)cc(F)c(F)c1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA4 P22748 2/20 0.44
TDP1 Q9NUW8 4/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
PKM P14618 1/20 0.35
CASP6 P55212 1/20 0.34
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
CTDSP1 Q9GZU7 1/20 0.34
CYP1A2 P05177 2/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
TP53 P04637 1/20 0.33
GRIN2D O15399 1/20 0.33
GRIN3B O60391 1/20 0.33
GRIN1 Q05586 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17080253 0.85 CA1 (0.39) CA1CA2CA4TDP1L3MBTL1
SCHEMBL29007693 0.84 CA1 (0.42) CA1CA2CA4TDP1L3MBTL1
SCHEMBL1994831 0.80 TDP1 (0.41) CA1CA2CA4TDP1ALDH1A1
SCHEMBL2687218 0.78 PKM (0.41) CA1CA2CA4TDP1PKM
SCHEMBL17042427 0.77 GPR35 (0.36) CA1CA2CA4TDP1L3MBTL1
SCHEMBL30515532 0.77 ALDH1A1 (0.41) CA1CA2TDP1L3MBTL1CASP6
SCHEMBL6217472 0.77 ALDH1A1 (0.41) CA1CA2TDP1L3MBTL1CASP6
SCHEMBL8872949 0.76 TDP1 (0.35) CA1CA2TDP1L3MBTL1PKM
SCHEMBL8161795 0.76 GPR35 (0.47) CA1CA2TDP1KDM4ECYP1A2
SCHEMBL2008253 0.75 CA1 (0.55) CA1CA2TDP1KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1304329-B1 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI SANKYO CO LTD (JP) 2008-10-15 EP disclosed
EP-0807630-B1 HETEROCYCLIC COMPOUNDS DAIICHI SEIYAKU CO (JP) 2003-05-07 EP disclosed
EP-1304329-A2 Pyridonecarboxylic acid derivatives and their use as antibacterial agents DAIICHI PHARMACEUTICAL CO., LTD. (JP) 2003-04-23 EP disclosed
US-5849757-A Pyridonecarboxylic acid derivatives substituted by a bicyclic amino group as antibacterials DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1998-12-15 US disclosed
EP-0807630-A1 HETEROCYCLIC COMPOUNDS DAIICHI PHARMACEUTICAL CO., LTD. (JP) 1997-11-19 EP disclosed
EP-0545866-A1 Process for the preparation of trifluorobenzol derivatives CIBA-GEIGY AG (CH) 1993-06-09 EP disclosed
EP-0545866-A1 Process for the preparation of trifluorobenzol derivatives CIBA-GEIGY AG (CH) 1993-06-09 EP disclosed